SCHEMBL20428776

SCHEMBL20428776

CSc1nc(-c2ccc(Cl)nc2)nn1COCCS(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 6/20 0.35
KMT2A Q03164 6/20 0.34
MAPT P10636 4/20 0.34
F2 P00734 2/20 0.34
HSD17B10 Q99714 2/20 0.34
TSHR P16473 2/20 0.34
TP53 P04637 1/20 0.34
NPC1 O15118 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
ACHE P22303 2/20 0.32
LIPE Q05469 2/20 0.32
GAA P10253 1/20 0.32
KLK7 P49862 1/20 0.32
KLK14 Q9P0G3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16661210 0.85 DGAT1 (0.38) RAB9AKDM4EALDH1A1NPSR1POLB
SCHEMBL18552799 0.84 RAB9A (0.35) RAB9AKDM4EALDH1A1NPSR1POLB
SCHEMBL18552801 0.82 PTGS2 (0.31) KDM4EALDH1A1POLBHPGDKMT2A
SCHEMBL16661275 0.81 PDE10A (0.34)
SCHEMBL20428575 0.77 MEN1 (0.37) KDM4EALDH1A1HPGDKMT2AMEN1
SCHEMBL16661257 0.75 DGAT1 (0.38) RAB9AKDM4EALDH1A1NPSR1POLB
SCHEMBL16660951 0.74 KDM4E (0.31) KDM4EALDH1A1HPGDMAPT
SCHEMBL18531176 0.73 CYP2A6 (0.33) RAB9AKMT2ANPC1MEN1
SCHEMBL20428777 0.72 PTGS2 (0.33) RAB9AKDM4EALDH1A1NPSR1POLB
SCHEMBL16660946 0.70 DGAT1 (0.39) RAB9AKDM4EPOLBSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2862856-B1 IMIDAZOLE AND TRIAZOLE COMPOUNDS AS DGAT-1 INHIBITORS MITSUBISHI TANABE PHARMA CORP (JP) 2018-08-01 EP disclosed