SCHEMBL2044587

SCHEMBL2044587

CN(C)C(=C(C=O)c1ccnc(Cl)c1)c1ccc(Cl)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.43
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
KMT2A Q03164 5/20 0.38
MEN1 O00255 3/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
HPGD P15428 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
ALOX12 P18054 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
F2 P00734 1/20 0.33
MAPK1 P28482 1/20 0.33
DAO P14920 1/20 0.33
TSHR P16473 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2044451 0.84 ALDH1A1 (0.43) ALDH1A1KDM4EGAAKMT2AMEN1
SCHEMBL2043622 0.75 ALDH1A1 (0.40) ALDH1A1KDM4EGAAKMT2AMEN1
SCHEMBL2044585 0.74 ALDH1A1 (0.46) ALDH1A1KDM4EGAAKMT2AMEN1
SCHEMBL2053724 0.74 ALDH1A1 (0.46) ALDH1A1KDM4EGAAKMT2AMEN1
SCHEMBL9111206 0.68 CYP11B1 (0.41) CYP11B1CYP11B2LMNATAS1R3TAS1R1
SCHEMBL4926597 0.67 TAS1R3 (0.44) ALDH1A1KMT2ACYP11B1CYP11B2HPGD
SCHEMBL27320783 0.64 POLB (0.38) CYP11B1CYP11B2TAS1R3TAS1R1TAS1R2
SCHEMBL6617730 0.63 F2 (0.59) ALDH1A1KDM4EGAAKMT2AMEN1
SCHEMBL2042913 0.62 GSK3B (0.50) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL17320231 0.61 HTT (0.61) ALDH1A1KDM4EGAAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2516423-A1 THIENYLPYRI (MI) DINYLAZOLE AND THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI Bayer CropScience AG (DE) 2012-10-31 EP disclosed
WO-2011076725-A1 THIENYLPYRI (MI) DINYLAZOLE AND THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI BAYER CROPSCIENCE AG (DE) 2011-06-30 WO disclosed