SCHEMBL20458152

SCHEMBL20458152

OC(Nc1nsc(-c2ccccc2)n1)[C@@H]1CCN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
TP53 P04637 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HTT P42858 5/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 1/20 0.41
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
NPY5R Q15761 1/20 0.34
RECQL P46063 1/20 0.34
CASR P41180 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20458153 0.77 ADORA3 (0.49) TP53HSD17B10HTTNPC1RAB9A
SCHEMBL9892932 0.74 KDM4E (0.53) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL20458212 0.72 RAB9A (0.50) KDM4EHTTNPC1RAB9ASMN1; SMN2
SCHEMBL16253075 0.68 KDM4E (0.49) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL13257156 0.68 KDM4E (0.49) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL3266075 0.63 TP53 (0.56) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL13842699 0.63 KDM4E (0.63) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL20458204 0.63 KDM4E (0.56) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL7656935 0.63 KDM4E (0.63) KDM4ETP53HSD17B10HTTNPC1
SCHEMBL9892890 0.63 HTT (0.60) KDM4ETP53HSD17B10HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443107-B1 AZETIDINE 2 -CARBOXAMIDE DERIVATIVES WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INT (DE) 2018-08-08 EP disclosed