SCHEMBL20460269

SCHEMBL20460269

COc1cccc2c(CN3CCOCC3)ccnc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.53
L3MBTL1 Q9Y468 4/20 0.53
PAX8 Q06710 2/20 0.53
NPC1 O15118 2/20 0.53
HTT P42858 8/20 0.52
SMN1; SMN2 Q16637 7/20 0.52
LMNA P02545 7/20 0.52
MAPT P10636 6/20 0.52
NPSR1 Q6W5P4 3/20 0.52
MPI P34949 2/20 0.52
NFKB1 P19838 2/20 0.52
NFKB2 Q00653 2/20 0.52
RELA Q04206 2/20 0.52
ALOX12 P18054 1/20 0.52
KMT2A Q03164 1/20 0.52
METAP2 P50579 1/20 0.50
TP53 P04637 5/20 0.49
KDM4E B2RXH2 5/20 0.49
TDP1 Q9NUW8 3/20 0.49
MAPK1 P28482 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28514468 0.78 PRKDC (0.52) NPC1LMNAMAPTKMT2ATP53
SCHEMBL20460320 0.77 KDM4E (0.67) RAB9AL3MBTL1PAX8NPC1HTT
SCHEMBL20460271 0.76 KDM4E (0.65) NPC1HTTSMN1; SMN2LMNAMAPT
SCHEMBL12530876 0.76 METAP2 (0.54) RAB9AL3MBTL1PAX8NPC1HTT
SCHEMBL31428721 0.76 ALDH1A1 (0.69) RAB9AL3MBTL1PAX8NPC1SMN1; SMN2
SCHEMBL23714056 0.75 L3MBTL1 (0.59) RAB9AL3MBTL1PAX8NPC1HTT
SCHEMBL16964453 0.75 HTR1A (0.60) RAB9AL3MBTL1NPC1HTTSMN1; SMN2
SCHEMBL14514792 0.75 CYP2A13 (0.63) L3MBTL1KMT2AKDM4EDRD2DRD4
SCHEMBL24716123 0.75 POLB (0.59) RAB9AL3MBTL1PAX8NPC1HTT
SCHEMBL30626612 0.75 POLB (0.59) RAB9AL3MBTL1PAX8NPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2288351-B1 NOVEL PYRROLIDONE DERIVATIVES FOR USE AS METAP-2 INHIBITORS MERCK PATENT GMBH (DE) 2018-08-08 EP disclosed