SCHEMBL2049474

SCHEMBL2049474

Fc1cccc(F)c1-c1[c]cccc1C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.36
HSD11B1 P28845 1/20 0.36
PTPN1 P18031 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
PDK2 Q15119 2/20 0.31
KCNN4 O15554 1/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17514475 0.86
SCHEMBL11302129 0.83 HSD11B1 (0.30) HSD11B1
SCHEMBL17514835 0.83 HSD11B1 (0.33) HSD11B1
SCHEMBL17515018 0.83 CYP11B1 (0.32)
SCHEMBL2049471 0.81 HSD11B1 (0.46) TRPA1HSD11B1PDK2KCNN4
SCHEMBL2437985 0.80 HSD11B1 (0.38) TRPA1HSD11B1SLC22A12PDK2KCNN4
SCHEMBL17514464 0.79 KIF11 (0.41) SLC22A12
SCHEMBL30568365 0.75 TRPA1 (0.47) TRPA1HSD11B1PTPN1SLC22A12PDK2
SCHEMBL2433532 0.74 NR1H2 (0.35)
SCHEMBL2426847 0.74 CYP11B2 (0.43) PTPN1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed