SCHEMBL20511447

SCHEMBL20511447

Clc1nc(Cl)nc(NCc2ccccc2Cl)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
PDE2A O00408 1/20 0.50
TP53 P04637 1/20 0.50
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
PDE5A O76074 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
CHRM2 P08172 1/20 0.47
PNMT P11086 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KCNN3 Q9UGI6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3788149 0.82 CD38 (0.46) TSHRPDE2ACYP3A4CYP2C19HSD17B10
SCHEMBL20511207 0.81 DCTPP1 (0.52) TSHRCHRM2KCNN3NFKB1MAPK1
SCHEMBL14869738 0.81 HRH4 (0.53) TP53HDAC3HDAC1HDAC2HDAC6
SCHEMBL20511040 0.79 HDAC3 (0.49) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL5477205 0.78 NPC1 (0.49) ALDH1A1POLBNPC1RAB9ACYP3A4
SCHEMBL6739809 0.78 GAA (0.58) TSHRTP53HDAC3HDAC1HDAC2
SCHEMBL1562297 0.76 APP (0.59) ALDH1A1PDE5ANFKB1GAAMAPT
SCHEMBL29558335 0.76 PDE5A (0.61) PDE2ATP53ALDH1A1POLBPDE5A
SCHEMBL6690806 0.75 RAB9A (0.67) TP53NPC1RAB9ACHRM2PNMT
SCHEMBL29168139 0.75 P2RX7 (0.46) TP53ALDH1A1POLBCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020146779-A1 mTORC1 INHIBITORS FOR ACTIVATING AUTOPHAGY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-07-16 WO disclosed
WO-2018175958-A1 THIOREDOXIN MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-09-27 WO disclosed