SCHEMBL20522882

SCHEMBL20522882

CCCCOC(=O)N1CCC(c2ccc(N)c(OC)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.56
QDPR P09417 2/20 0.49
HTR4 Q13639 4/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
ADRA2C P18825 1/20 0.47
CHRM3 P20309 1/20 0.47
HTR1D P28221 1/20 0.47
ADRA1B P35368 1/20 0.47
HTR2B P41595 1/20 0.47
HTR3A P46098 1/20 0.47
PDE4A P27815 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
TRPC6 Q9Y210 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345819 0.91 PDE4B (0.56) PDE4BQDPRPDE4APDE4CPDE4D
SCHEMBL3639005 0.83 QDPR (0.50) PDE4BQDPRPDE4APDE4CPDE4D
SCHEMBL30376364 0.83 LMNA (0.49) PDE4BCHRM4PDE4DCHRM2CHRM1
SCHEMBL13362111 0.82 QDPR (0.55) PDE4BQDPRPDE4APDE4CPDE4D
SCHEMBL22659030 0.80 PDE4B (0.53) PDE4BPDE4APDE4CPDE4D
SCHEMBL25260521 0.80 MAPT (0.49) HTR4CHRM4CHRM5ADRA2CCHRM3
SCHEMBL2227613 0.80 QDPR (0.59) PDE4BQDPRPDE4APDE4CPDE4D
SCHEMBL3311407 0.80 QDPR (0.74) PDE4BQDPRPDE4APDE4CPDE4D
SCHEMBL520443 0.80 QDPR (0.53) PDE4BQDPR
SCHEMBL310046 0.80 PDE4B (0.62) PDE4BQDPRPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600327-A1 HETEROCYCLIC COMPOUND Cardurion Pharmaceuticals, LLC (US) 2020-02-05 EP disclosed
WO-2018183112-A1 HETEROCYCLIC COMPOUND CARDURION PHARMACEUTICALS, LLC (US) 2018-10-04 WO disclosed