SCHEMBL20524610

SCHEMBL20524610

Cc1cnc(N2CCN(C(=O)O)CC2)c(N)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMO Q99835 4/20 0.38
OPRK1 P41145 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 2/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.35
HPGD P15428 1/20 0.35
P2RY12 Q9H244 4/20 0.35
HRH4 Q9H3N8 1/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20524606 0.82 OPRK1 (0.41) OPRK1KDM4ELMNAMAPTALDH1A1
SCHEMBL22712188 0.81 KIT (0.48) MEN1KMT2ALMNAMAPTALDH1A1
SCHEMBL30323222 0.81 KIT (0.48) MEN1KMT2ALMNAMAPTALDH1A1
SCHEMBL27741477 0.79 OPRK1 (0.39) OPRK1MEN1KMT2AKDM4ELMNA
SCHEMBL3434342 0.79 MEN1 (0.40) OPRK1MEN1KMT2ALMNATP53
SCHEMBL13106057 0.78 MDM2 (0.44) OPRK1LMNATP53
SCHEMBL20524637 0.78 ALDH1A1 (0.49) OPRK1LMNAMAPTALDH1A1
SCHEMBL27848265 0.74 ALDH1A1 (0.47) SMOLMNATP53MAPTALDH1A1
SCHEMBL16178191 0.73 SMO (0.43) SMOMEN1KMT2AKDM4ELMNA
SCHEMBL27741480 0.73 SMN1; SMN2 (0.46) MEN1KMT2ALMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600312-A1 PIPERIDINYL- AND PIPERAZINYL-SUBSTITUTED HETEROAROMATIC CARBOXAMIDES AS MODULATORS OF GPR6 Takeda Pharmaceutical Company Limited (JP) 2020-02-05 EP disclosed
WO-2018183145-A1 PIPERIDINYL- AND PIPERAZINYL-SUBSTITUTED HETEROAROMATIC CARBOXAMIDES AS MODULATORS OF GPR6 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-10-04 WO disclosed