SCHEMBL20524637

SCHEMBL20524637

Cc1cnc(N2CCN(C(=O)O)CC2)c([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
MAPK1 P28482 2/20 0.49
HTT P42858 2/20 0.49
POLB P06746 2/20 0.44
OPRK1 P41145 1/20 0.43
GRM5 P41594 2/20 0.43
LMNA P02545 4/20 0.42
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
HSD11B1 P28845 1/20 0.40
MAPT P10636 1/20 0.40
JAK2 O60674 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30323135 0.83 MAPT (0.53) ALDH1A1MAPK1HTTPOLBOPRK1
SCHEMBL22712080 0.83 MAPT (0.53) ALDH1A1MAPK1HTTPOLBOPRK1
SCHEMBL29274197 0.81 SMN1; SMN2 (0.48) ALDH1A1MAPK1HTTPOLBLMNA
SCHEMBL20524655 0.81 OPRK1 (0.44) ALDH1A1MAPK1HTTOPRK1GRM5
SCHEMBL3435982 0.80 ALDH1A1 (0.45) ALDH1A1MAPK1HTTPOLBOPRK1
SCHEMBL4606448 0.79 ALDH1A1 (0.49) ALDH1A1MAPK1HTTOPRK1LMNA
SCHEMBL20524610 0.78 SMO (0.38) ALDH1A1OPRK1LMNAMAPT
SCHEMBL3435641 0.77 ALDH1A1 (0.50) ALDH1A1MAPK1HTTPOLBOPRK1
SCHEMBL16178366 0.76 ALDH1A1 (0.66) ALDH1A1MAPK1HTTLMNASMN1; SMN2
SCHEMBL6949066 0.76 MAPK1 (0.49) ALDH1A1MAPK1HTTPOLBGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600312-A1 PIPERIDINYL- AND PIPERAZINYL-SUBSTITUTED HETEROAROMATIC CARBOXAMIDES AS MODULATORS OF GPR6 Takeda Pharmaceutical Company Limited (JP) 2020-02-05 EP disclosed
WO-2018183145-A1 PIPERIDINYL- AND PIPERAZINYL-SUBSTITUTED HETEROAROMATIC CARBOXAMIDES AS MODULATORS OF GPR6 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-10-04 WO disclosed