SCHEMBL2052473

SCHEMBL2052473

OC1COC(c2nccs2)OC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
NOS1 P29475 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20789355 0.79 ADORA3 (0.31) NOS3NOS2
SCHEMBL4770134 0.77 KIF11 (0.36) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL2053635 0.74 NOS3 (0.35) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL21178116 0.73 DRD4 (0.40) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL21178152 0.73 DRD4 (0.40) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL21178115 0.73 DRD4 (0.40) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL2014387 0.71 ALDH1A1 (0.34) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL24676709 0.70 DRD4 (0.36) NOS3NOS2ALDH1A1TSHRNOS1
SCHEMBL2043681 0.69 KIF11 (0.31)
SCHEMBL28089091 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513098-A1 AMINOPYRIMIDINES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-10-24 EP disclosed
WO-2011075515-A1 AMINOPYRIMIDINES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed