SCHEMBL20525337

SCHEMBL20525337

CC(C)(C)CN1CCC(c2ccnc3c2ccn3Cc2ccc(C(N)=O)c(O)c2)CC1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 1/20 0.34
FGFR4 P22455 1/20 0.34
PARP1 P09874 2/20 0.34
DRD2 P14416 1/20 0.34
HTR6 P50406 1/20 0.34
PARP2 Q9UGN5 1/20 0.33
CAMKK1 Q8N5S9 1/20 0.33
CAMKK2 Q96RR4 1/20 0.33
SYK P43405 6/20 0.32
KCNH2 Q12809 2/20 0.32
P2RY1 P47900 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
HTR4 Q13639 2/20 0.31
ACHE P22303 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525467 0.94 FGFR1 (0.34) FGFR1FGFR4DRD2HTR6CAMKK1
SCHEMBL20525360 0.87 PARP1 (0.39) FGFR1FGFR4PARP1DRD2HTR6
SCHEMBL20525552 0.87 DRD2 (0.36) FGFR1FGFR4PARP1DRD2HTR6
SCHEMBL20525429 0.86 CHUK (0.39) FGFR1FGFR4PARP1DRD2HTR6
SCHEMBL20525349 0.84 SCN9A (0.46) PARP1PARP2KCNH2SCN5ASCN9A
SCHEMBL20525347 0.84 JAK1 (0.47) DRD2SYK
SCHEMBL20525434 0.83 OPRM1 (0.35) FGFR1FGFR4CAMKK1CAMKK2SYK
SCHEMBL18108920 0.80 HDAC6 (0.45) KCNH2
SCHEMBL16804352 0.80 KDM4E (0.41) KCNH2P2RY1
SCHEMBL16804244 0.77 JAK2 (0.41) FGFR1FGFR4DRD2HTR6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed