SCHEMBL20525347

SCHEMBL20525347

COc1cccc(CN2CCC(c3ccnc4c3ccn4Cc3ccc(C(N)=O)c(O)c3)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.47
FAAH O00519 1/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
MAPT P10636 1/20 0.43
DRD4 P21917 1/20 0.42
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
JAK3 P52333 2/20 0.40
JAK2 O60674 1/20 0.40
TYK2 P29597 1/20 0.40
POLB P06746 1/20 0.40
SYK P43405 1/20 0.40
ADRA1D P25100 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
GAA P10253 1/20 0.40
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525349 0.87 SCN9A (0.46) JAK1KDM4EDRD4JAK3JAK2
SCHEMBL20525360 0.86 PARP1 (0.39) DRD2
SCHEMBL20525552 0.86 DRD2 (0.36) SYKDRD2
SCHEMBL20525428 0.86 KDM4E (0.47) JAK1KDM4EALDH1A1DRD4KLKB1
SCHEMBL18109017 0.85 LMNA (0.50) FAAHKDM4EALDH1A1MAPTDRD4
SCHEMBL20525429 0.85 CHUK (0.39) JAK2TYK2SYKDRD2
SCHEMBL20525337 0.84 FGFR1 (0.34) SYKDRD2
SCHEMBL16804168 0.84 HDAC1 (0.50) FAAHKDM4EALDH1A1MAPTDRD4
SCHEMBL20525467 0.83 FGFR1 (0.34) SYKDRD2
SCHEMBL20525475 0.83 JAK1 (0.47) JAK1FAAHKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed