SCHEMBL20525428

SCHEMBL20525428

COc1cccc(CN2CCN(c3ccnc4c3ccn4Cc3ccc(C(N)=O)c(O)c3)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.47
JAK1 P23458 1/20 0.43
KLKB1 P03952 1/20 0.43
KLK1 P06870 1/20 0.43
DRD2 P14416 5/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
HTR6 P50406 4/20 0.42
GPR52 Q9Y2T5 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
ADRA1D P25100 1/20 0.41
SRPK1 Q96SB4 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525353 0.93 HDAC1 (0.41) ALDH1A1GAAKLKB1KLK1DRD2
SCHEMBL20525423 0.86 SCN9A (0.42) KDM4EALDH1A1DRD2DRD4DRD3
SCHEMBL20525347 0.86 JAK1 (0.47) KDM4EALDH1A1GAAJAK1KLKB1
SCHEMBL20525447 0.86 HTR6 (0.41) KDM4EALDH1A1DRD2HTR6SRPK1
SCHEMBL18108845 0.85 LMNA (0.51) KDM4EALDH1A1GAAKLKB1KLK1
SCHEMBL20525329 0.84 GHSR (0.43) ALDH1A1JAK1
SCHEMBL16804340 0.83 HDAC1 (0.53) KDM4EALDH1A1GAAKLKB1KLK1
SCHEMBL20525472 0.83 CYP3A4 (0.40) ALDH1A1JAK1MEN1KMT2A
SCHEMBL20525448 0.83 RPS6KB1 (0.41) KDM4EALDH1A1DRD2HTR6SRPK1
SCHEMBL20525450 0.81 F12 (0.36) DRD2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed