SCHEMBL20525447

SCHEMBL20525447

NC(=O)c1ccc(Cn2ccc3c(N4CCN(Cc5ccncc5)CC4)ccnc32)cc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.41
DRD2 P14416 4/20 0.41
SCN9A Q15858 1/20 0.38
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CDC7 O00311 1/20 0.36
CDK9 P50750 1/20 0.36
FGFR1 P11362 1/20 0.35
FGFR4 P22455 1/20 0.35
CTSB P07858 1/20 0.35
PARP1 P09874 1/20 0.35
SRPK1 Q96SB4 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
ALDH1A1 P00352 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525448 0.91 RPS6KB1 (0.41) HTR6DRD2SCN9APARP1SRPK1
SCHEMBL20525353 0.90 HDAC1 (0.41) HTR6DRD2ALDH1A1
SCHEMBL20525423 0.90 SCN9A (0.42) HTR6DRD2SCN9ACA12CA1
SCHEMBL20525428 0.86 KDM4E (0.47) HTR6DRD2SRPK1ALDH1A1KDM4E
SCHEMBL20525450 0.85 F12 (0.36) HTR6DRD2FGFR1FGFR4PARP1
SCHEMBL20525329 0.81 GHSR (0.43) ALDH1A1
SCHEMBL20525382 0.81 CYP1A2 (0.38) HTR6DRD2SCN9APARP1ALDH1A1
SCHEMBL20525430 0.80 PARP1 (0.41) HTR6DRD2FGFR1FGFR4PARP1
SCHEMBL20525346 0.80 SMN1; SMN2 (0.43) PARP1ALDH1A1KDM4E
SCHEMBL18108947 0.80 HDAC1 (0.48) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed