SCHEMBL20525448

SCHEMBL20525448

NC(=O)c1ccc(Cn2ccc3c(N4CCN(Cc5ccc(C(F)(F)F)cc5)CC4)ccnc32)cc1O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 3/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
DRD2 P14416 4/20 0.40
HTR6 P50406 4/20 0.40
SRPK1 Q96SB4 4/20 0.39
ACHE P22303 1/20 0.39
HIF1A Q16665 1/20 0.38
EPAS1 Q99814 1/20 0.38
CASP1 P29466 1/20 0.38
CASP4 P49662 1/20 0.38
CASP5 P51878 1/20 0.38
AKT1 P31749 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525447 0.91 HTR6 (0.41) KDM4EALDH1A1PARP1DRD2HTR6
SCHEMBL20525346 0.89 SMN1; SMN2 (0.43) RPS6KB1KDM4EALDH1A1SMN1; SMN2PARP1
SCHEMBL20525353 0.87 HDAC1 (0.41) ALDH1A1DRD2HTR6MAPT
SCHEMBL20525423 0.85 SCN9A (0.42) KDM4EALDH1A1PARP1PARP2DRD2
SCHEMBL20525430 0.84 PARP1 (0.41) RPS6KB1PARP1DRD2HTR6AKT1
SCHEMBL18108960 0.83 HIF1A (0.47) KDM4EALDH1A1SRPK1ACHEHIF1A
SCHEMBL20525428 0.83 KDM4E (0.47) KDM4EALDH1A1DRD2HTR6SRPK1
SCHEMBL20525450 0.82 F12 (0.36) RPS6KB1PARP1PARP2DRD2HTR6
SCHEMBL18108967 0.82 HIF1A (0.50) SRPK1ACHEHIF1AEPAS1
SCHEMBL20525410 0.81 ENPP2 (0.36) RPS6KB1DRD2HTR6AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed