SCHEMBL20525346

SCHEMBL20525346

NC(=O)c1ccc(Cn2ccc3c(N4CCN(c5ccc(C(F)(F)F)cn5)CC4)ccnc32)cc1O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.43
KDM4E B2RXH2 6/20 0.43
LMNA P02545 3/20 0.43
HTT P42858 2/20 0.43
PARP1 P09874 3/20 0.42
ABL1 P00519 1/20 0.41
TIPARP Q7Z3E1 1/20 0.40
RPS6KB1 P23443 2/20 0.40
HPGD P15428 1/20 0.40
ALDH1A1 P00352 1/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
MAPT P10636 2/20 0.38
AKT1 P31749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525430 0.89 PARP1 (0.41) PARP1RPS6KB1AKT1
SCHEMBL20525448 0.89 RPS6KB1 (0.41) SMN1; SMN2KDM4EPARP1RPS6KB1ALDH1A1
SCHEMBL18108887 0.82 MAPT (0.45) SMN1; SMN2KDM4ELMNAHTTHPGD
SCHEMBL20525450 0.81 F12 (0.36) PARP1RPS6KB1
SCHEMBL18108893 0.80 SMN1; SMN2 (0.46) SMN1; SMN2KDM4ELMNAHTTHPGD
SCHEMBL20525447 0.80 HTR6 (0.41) KDM4EPARP1ALDH1A1
SCHEMBL20525410 0.79 ENPP2 (0.36) RPS6KB1JAK2AKT1
SCHEMBL20525423 0.79 SCN9A (0.42) KDM4EPARP1ALDH1A1
SCHEMBL20525353 0.77 HDAC1 (0.41) LMNAALDH1A1MAPT
SCHEMBL20525344 0.75 DRD2 (0.33) AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed