SCHEMBL2053317

SCHEMBL2053317

Fc1ccc(-c2cc[c]c(C(F)(F)F)c2)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
DHFR P00374 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
LMNA P02545 1/20 0.42
ALB P02768 1/20 0.42
HMGB1 P09429 1/20 0.42
HPGD P15428 1/20 0.42
CXCL12 P48061 1/20 0.42
KMT2A Q03164 1/20 0.42
HIF1A Q16665 1/20 0.42
SLC22A6 Q4U2R8 1/20 0.42
ACMSD Q8TDX5 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP2 O95551 1/20 0.39
ALOX5AP P20292 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2050766 0.87 TRPA1 (0.32) TRPA1PDE3BPDE3A
SCHEMBL15637441 0.83 ESR1 (0.30) ESR1ESR2
SCHEMBL2431244 0.81 PDK2 (0.42) ACMSDALOX5APFEN1TRPA1
SCHEMBL15637425 0.80 GABRA1 (0.39) ALOX5APFEN1
SCHEMBL2431524 0.79 PDK2 (0.35) KDM4E
SCHEMBL436196 0.79 TTR (0.46) TTRKDM4EMEN1USP2ALDH1A1
SCHEMBL5261997 0.77 PDK2 (0.40) MEN1HPGDKMT2ATDP2CNR1
SCHEMBL432713 0.76 TTR (0.44) TTRKDM4EMEN1USP2ALDH1A1
SCHEMBL15637656 0.76 TTR (0.44) TTRKDM4EMEN1USP2ALDH1A1
SCHEMBL2053488 0.76 ALDH1A1 (0.44) TTRKDM4EMEN1USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903440-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer CropScience AG (DE) 2015-08-12 EP disclosed
WO-2014053450-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2014-04-10 WO disclosed
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed