SCHEMBL20534680

SCHEMBL20534680

CC(CCC(=O)O)c1c(F)cccc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGFR P43088 3/20 0.43
PTGS2 P35354 1/20 0.40
EPHX2 P34913 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
CTSA P10619 1/20 0.37
CTSS P25774 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
FFAR4 Q5NUL3 2/20 0.36
FFAR1 O14842 1/20 0.36
RORC P51449 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20535701 0.86 FFAR4 (0.43) PTGFRSMN1; SMN2FFAR4
SCHEMBL21631962 0.81 PTGFR (0.46) PTGFRPTGS2CTSAFFAR4FFAR1
SCHEMBL21632087 0.80 PTGFR (0.39) PTGFRPTGS2EPHX2CTSACTSS
SCHEMBL20534568 0.79 KDM4E (0.42) PTGFRPTGS2SMN1; SMN2FFAR4
SCHEMBL20536700 0.78 CNR2 (0.47) PTGFREPHX2SMN1; SMN2FFAR4FFAR1
SCHEMBL19405291 0.77 CTSS (0.40) PTGS2AKR1C3AKR1C2CTSSSLC6A2
SCHEMBL20534638 0.75 KMT2A (0.41) SMN1; SMN2FFAR4FFAR1
SCHEMBL24106022 0.73 P2RX7 (0.40) EPHX2CTSS
SCHEMBL20534596 0.73 FFAR4 (0.41) PTGFRFFAR4FFAR1
SCHEMBL4547921 0.72 P2RX7 (0.42) PTGS2AKR1C3AKR1C2CTSSSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609870-A1 SUBSTITUTED N-ARYLETHYL-2-AMINOQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed
WO-2018189012-A1 SUBSTITUTED N-ARYLETHYL-2-AMINOQUINOLINE-4-CARBOXAMIDES AND USE THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2018-10-18 WO disclosed