SCHEMBL20534820

SCHEMBL20534820

NC(=O)c1oc2ccc(-c3ccc(C(F)(F)F)cc3)cc2c1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.56
ALDH1A1 P00352 5/20 0.56
HPGD P15428 4/20 0.56
HSD17B10 Q99714 4/20 0.56
IKBKB O14920 1/20 0.45
DHODH Q02127 1/20 0.43
KIF11 P52732 4/20 0.43
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C8 P10632 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP4B1 P13584 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP3A5 P20815 1/20 0.40
CYP2A7 P20853 1/20 0.40
CYP3A7 P24462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20534970 0.89 ALDH1A1 (0.46) KDM4EALDH1A1HPGDHSD17B10IKBKB
SCHEMBL20535692 0.88 KDM4E (0.52) KDM4EALDH1A1HPGDHSD17B10DHODH
SCHEMBL20535965 0.85 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10IKBKB
SCHEMBL20535680 0.83 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL20535044 0.83 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10IKBKB
SCHEMBL20535014 0.82 KDM4E (0.78) KDM4EALDH1A1HPGDHSD17B10IKBKB
SCHEMBL20535672 0.82 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL13699689 0.80 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10IKBKB
SCHEMBL20535529 0.80 ALDH1A1 (0.51) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL20534973 0.79 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018189683-A1 BENZOFURAN DERIVATIVES FOR USE AS AMPK ACTIVATORS UNIVERSITA' DI PISA (IT) 2018-10-18 WO claimed
WO-2018189683-A1 BENZOFURAN DERIVATIVES FOR USE AS AMPK ACTIVATORS UNIVERSITA' DI PISA (IT) 2018-10-18 WO disclosed