SCHEMBL2053792

SCHEMBL2053792

Fc1ccc(-c2cc[c]cc2C(F)(F)F)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
AR P10275 5/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
IDO1 P14902 2/20 0.33
TRPA1 O75762 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
DPP4 P27487 1/20 0.31
HSD11B1 P28845 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PLK4 O00444 1/20 0.30
AURKA O14965 1/20 0.30
MAPK13 O15264 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2052768 0.87 PDE3B (0.39) PDE3BPDE3AGLAPOLBGAA
SCHEMBL17514846 0.84 HSD11B1 (0.43) GLAPOLBGAATSHRAR
SCHEMBL17514963 0.84 HSD11B1 (0.43) GLAPOLBGAATSHRAR
SCHEMBL436101 0.82 IDO1 (0.38) PDE3BPDE3AIDO1DPP4ALDH1A1
SCHEMBL14483362 0.82 GLA (0.38) GLAPOLBGAATSHR
SCHEMBL17514477 0.81 AR (0.30) AR
SCHEMBL1274101 0.80 KIF11 (0.40) PDE3BPDE3AAKR1C3AKR1C2
SCHEMBL2437987 0.79 PDE3B (0.36) PDE3BPDE3AARAKR1C3AKR1C2
SCHEMBL2433534 0.77 PDE3B (0.36) PDE3BPDE3APOLBGAAAR
SCHEMBL2013845 0.76 AR (0.32) ARTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed