SCHEMBL205608

SCHEMBL205608

Fc1cccc(Cc2cs[c]n2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.40
IDO1 P14902 2/20 0.39
AGXT P21549 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
DAO P14920 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
BRD4 O60885 1/20 0.36
P2RX7 Q99572 1/20 0.36
MIF P14174 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
MPO P05164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1255674 0.72 MPO (0.36) MPO
SCHEMBL3300303 0.72 TAAR1 (0.60) TAAR1IDO1AGXTALDH1A1DAO
SCHEMBL17028856 0.69 HSP90AB1 (0.42) TAAR1IDO1MEN1KMT2AALDH1A1
SCHEMBL2092840 0.69 CA2 (0.56) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL4212164 0.68 KDM4E (0.61) TAAR1IDO1AGXTMEN1KMT2A
SCHEMBL6050957 0.68 KDM4E (0.51) TAAR1IDO1MEN1KMT2AKDM4E
SCHEMBL6235370 0.68 IDO1 (0.42) TAAR1IDO1AGXTMEN1KMT2A
SCHEMBL28816893 0.67 NPC1 (0.50) TAAR1IDO1AGXTTLR8TLR7
SCHEMBL4677 0.67 TAAR1 (0.42) TAAR1IDO1AGXTKDM4EDAO
SCHEMBL3298408 0.67 CALM1 (0.57) TAAR1IDO1AGXTALDH1A1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088806-B2 Thiazole compounds and methods of use ACHILLION PHARMACEUTICALS, INC. (US) 2012-01-03 US disclosed