SCHEMBL20565243

SCHEMBL20565243

COC(=O)C[C@@H]1CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
PKM P14618 1/20 0.47
GLS O94925 4/20 0.46
EPHX1 P07099 1/20 0.46
NR1H2 P55055 1/20 0.46
HPGD P15428 1/20 0.44
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
USP30 Q70CQ3 1/20 0.43
BRD4 O60885 1/20 0.43
RECQL P46063 1/20 0.43
PTPN2 P17706 1/20 0.42
PTPN1 P18031 1/20 0.42
PTPN6 P29350 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL852498 1.00 KDM4E (0.47) KDM4EPKMGLSEPHX1NR1H2
SCHEMBL19511364 1.00 KDM4E (0.47) KDM4EPKMGLSEPHX1NR1H2
SCHEMBL1048156 0.92 GLS (0.54) GLSEPHX1NR1H2HPGDALDH1A1
SCHEMBL1048155 0.92 GLS (0.54) GLSEPHX1NR1H2HPGDALDH1A1
SCHEMBL30922668 0.92 GLS (0.54) GLSEPHX1NR1H2HPGDALDH1A1
SCHEMBL106242 0.91 KDM4E (0.52) KDM4EPKMGLSEPHX1NR1H2
SCHEMBL31189316 0.91 NR1H2 (0.48) KDM4EPKMGLSEPHX1NR1H2
SCHEMBL31588543 0.91 NR1H2 (0.48) KDM4EPKMGLSEPHX1NR1H2
SCHEMBL25957458 0.91 NR1H2 (0.48) KDM4EPKMGLSEPHX1NR1H2
Hydrochloric Acid SCHEMBL4219415 0.90 KDM4E (0.51) KDM4EPKMGLSEPHX1NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4692057-A1 NOVEL B0AT1 INHIBITOR Mitsubishi Tanabe Pharma Corporation (JP) 2026-02-11 EP disclosed
US-20260001849-A1 NOVEL B0AT1 INHIBITOR MITSUBISHI TANABE PHARMA CORPORATION (JP) 2026-01-01 US disclosed
US-20250230140-A1 NOVEL TRIAZOLE-PYRIDINE SUBSTITUTED PYRROLIDINYL AND TETRAHYDRO-2H-PYRANYL ACETIC ACID COMPOUNDS AS LPA ANTAGONISTS VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2025-07-17 US disclosed
WO-2024210198-A1 NOVEL B0AT1 INHIBITOR 田辺三菱製薬株式会社 2024-10-10 WO disclosed
CN-117751106-A Novel triazole-pyridine substituted pyrrolidinyl and tetrahydro-2H-pyranylacetic acid compounds as LPA antagonists 唯久生物技术(苏州)有限公司 2024-03-22 CN disclosed
EP-4330249-A1 NOVEL TRIAZOLE-PYRIDINE SUBSTITUTED PYRROLIDINYL AND TETRAHYDRO-2H-PYRANYL ACETIC ACID COMPOUNDS AS LPA ANTAGONISTS Viva Star Biosciences (Suzhou) Co., Ltd. (CN) 2024-03-06 EP disclosed
WO-2022232459-A1 NOVEL TRIAZOLE-PYRIDINE SUBSTITUTED PYRROLIDINYL AND TETRAHYDRO-2H-PYRANYL ACETIC ACID COMPOUNDS AS LPA ANTAGONISTS VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2022-11-03 WO disclosed
EP-3624797-A1 KINASE INHIBITORS AND USES THEREOF Denali Therapeutics Inc. (US) 2020-03-25 EP disclosed
WO-2018213632-A1 KINASE INHIBITORS AND USES THEREOF DENALI THERAPEUTICS INC. (US) 2018-11-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260001849-A1 NOVEL B0AT1 INHIBITOR BCAT1, BCAT2, BHMT KDM4E 3501/4885PKM 1042/4885GLS 77/4885
US-20250230140-A1 NOVEL TRIAZOLE-PYRIDINE SUBSTITUTED PYRROLIDINYL AND TETRAHYDRO-2H-PYRANYL ACETIC ACID COMPOUNDS AS LPA ANTAGONISTS LPAR3, LPAR2, LPAR1 KDM4E 3096/4885PKM 1629/4885GLS 1688/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.