SCHEMBL20568623

SCHEMBL20568623

Nc1nccc(Br)c1OCCCCl

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KLK1 P06870 1/20 0.34
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NOS3 P29474 3/20 0.31
NOS2 P35228 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19932671 0.93 NPC1 (0.32) KLK1NPC1HTTRAB9ASMN1; SMN2
SCHEMBL25385808 0.78 SMN1; SMN2 (0.42) HTTSMN1; SMN2NOS3NOS2
SCHEMBL31423975 0.74 ADORA2A (0.39) NPC1HTTRAB9ASMN1; SMN2NOS3
SCHEMBL3711280 0.73 ALOX5AP (0.41) HTTNOS3NOS2
SCHEMBL25228489 0.69 NOS2 (0.35) NOS3NOS2
SCHEMBL30731229 0.68 PTPN1 (0.35)
SCHEMBL7843486 0.67 LTA4H (0.56) NPC1HTTRAB9ASMN1; SMN2NOS3
SCHEMBL24568101 0.67 KLK1 (0.37) KLK1
SCHEMBL1796382 0.66 SMN1; SMN2 (0.35) KLK1NPC1RAB9ASMN1; SMN2
SCHEMBL18338657 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601752-A Novel inhibitors of MAP4K1 伊克诺斯科学公司 2021-04-02 CN disclosed
EP-3630778-A1 NOVEL INHIBITORS OF MAP4K1 Ichnos Sciences SA (CH) 2020-04-08 EP disclosed
WO-2018215668-A1 NOVEL INHIBITORS OF MAP4K1 GLENMARK PHARMACEUTICALS S.A. (CH) 2018-11-29 WO disclosed