SCHEMBL20569491

SCHEMBL20569491

O=[N+]([O-])c1cc(N2CCCNCC2)cc(C(F)(F)F)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.65
ADRB1 P08588 2/20 0.60
SIRT6 Q8N6T7 1/20 0.50
ALDH1A1 P00352 4/20 0.48
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR1D P28221 1/20 0.48
HTR2C P28335 1/20 0.48
HTR3A P46098 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
MAPT P10636 7/20 0.47
THRB P10828 1/20 0.47
HTR1A P08908 1/20 0.44
HTR7 P34969 1/20 0.44
MET P08581 1/20 0.43
MAPK1 P28482 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15542432 0.95 ADRB1 (0.67) SMN1; SMN2ADRB1SIRT6ALDH1A1HTR3E
Hydrochloric Acid SCHEMBL20568855 0.93 ADRB1 (0.65) SMN1; SMN2ADRB1SIRT6ALDH1A1HTR3E
SCHEMBL6562147 0.80 ADRB1 (0.69) SMN1; SMN2ADRB1SIRT6ALDH1A1HTR3E
SCHEMBL20567878 0.80 LMNA (0.59) SMN1; SMN2SIRT6ALDH1A1MAPTMET
SCHEMBL15542558 0.79 SLC6A9 (0.52) SMN1; SMN2ADRB1ALDH1A1MAPTMET
SCHEMBL15542522 0.79 CYP2C9 (0.46) SMN1; SMN2ADRB1ALDH1A1MAPTMEN1
SCHEMBL2972930 0.79 SIRT6 (0.55) ADRB1SIRT6ALDH1A1MAPTMET
SCHEMBL15553691 0.79 MAPT (0.55) SMN1; SMN2ADRB1ALDH1A1MAPTTHRB
SCHEMBL20568475 0.77 ADRB1 (0.42) SMN1; SMN2ADRB1MAPTMEN1KMT2A
SCHEMBL16895216 0.77 ADRB1 (0.42) SMN1; SMN2ADRB1SIRT6ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601752-A Novel inhibitors of MAP4K1 伊克诺斯科学公司 2021-04-02 CN disclosed
EP-3630778-A1 NOVEL INHIBITORS OF MAP4K1 Ichnos Sciences SA (CH) 2020-04-08 EP disclosed
WO-2018215668-A1 NOVEL INHIBITORS OF MAP4K1 GLENMARK PHARMACEUTICALS S.A. (CH) 2018-11-29 WO disclosed