SCHEMBL20591997

SCHEMBL20591997

O=C(O)c1ccc(-c2ccccc2)c(-c2ccc([N+](=O)[O-])cc2[N+](=O)[O-])c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.51
POLB P06746 2/20 0.50
CES2 O00748 2/20 0.50
RAB9A P51151 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TTR P02766 1/20 0.49
MAPK1 P28482 1/20 0.49
LMNA P02545 1/20 0.49
CASP6 P55212 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
PTGS2 P35354 2/20 0.48
MYC P01106 1/20 0.47
MAX P61244 1/20 0.47
MAPT P10636 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
HCAR3 P49019 1/20 0.46
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062366 0.87 CASP6 (0.64) TP53CES2MEN1KMT2ATTR
SCHEMBL11781006 0.84 TDP1 (0.61) TP53POLBCES2MEN1KMT2A
SCHEMBL11351696 0.84 ALDH1A1 (0.58) TP53POLBCES2RAB9AMEN1
SCHEMBL99918 0.84 CASP6 (0.64) POLBLMNACASP6TDP1MAPT
SCHEMBL2137404 0.82 ALDH1A1 (0.63) TP53POLBCES2RAB9AMAPK1
Water SCHEMBL27408458 0.81 ALDH1A1 (0.61) TP53POLBCES2RAB9AMAPK1
Formaldehyde SCHEMBL29219144 0.79 ALDH1A1 (0.59) TP53POLBCES2RAB9AMAPK1
SCHEMBL11195885 0.79 CASP6 (0.75) LMNACASP6HCAR3TSHR
Acrylamide SCHEMBL16586177 0.78 POLB (0.47) TP53POLBCES2RAB9AMEN1
Hydrochloric Acid SCHEMBL9784149 0.77 CASP6 (0.62) POLBTTRLMNACASP6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210255193-A1 LYSINE REACTIVE PROBES AND USES THEREOF THE SCRIPPS RESEARCH INSTITUTE 2021-08-19 US disclosed
EP-3642630-A1 LYSINE REACTIVE PROBES AND USES THEREOF The Scripps Research Institute (US) 2020-04-29 EP disclosed
WO-2018237334-A1 LYSINE REACTIVE PROBES AND USES THEREOF THE SCRIPPS RESEARCH INSTITUTE (US) 2018-12-27 WO disclosed
US-20180372751-A1 LYSINE REACTIVE PROBES AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2018-12-27 US disclosed