SCHEMBL20657355

SCHEMBL20657355

N#Cc1ccc(-c2cc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc3)no2)cc1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.62
POLB P06746 1/20 0.62
RXFP1 Q9HBX9 1/20 0.60
ACR P10323 1/20 0.57
TDP1 Q9NUW8 1/20 0.56
LMNA P02545 4/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
KDM4E B2RXH2 2/20 0.52
SCD O00767 1/20 0.51
MAPT P10636 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
GAA P10253 1/20 0.48
MAPKAPK2 P49137 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20657285 0.78 ALDH1A1 (0.64) ALDH1A1POLBTDP1LMNASMN1; SMN2
SCHEMBL1140233 0.76 CYP1A2 (0.60) ALDH1A1POLBTDP1LMNASMN1; SMN2
SCHEMBL1140302 0.76 MAPT (0.56) ALDH1A1POLBTDP1LMNAKDM4E
SCHEMBL1140119 0.76 MEN1 (0.60) ALDH1A1POLBTDP1LMNAKDM4E
SCHEMBL1140378 0.76 TDP1 (0.54) ALDH1A1POLBTDP1LMNAKDM4E
SCHEMBL8692256 0.76 ALDH1A1 (0.68) ALDH1A1POLBTDP1LMNASMN1; SMN2
SCHEMBL1140817 0.75 KMT2A (0.59) ALDH1A1POLBTDP1LMNASMN1; SMN2
SCHEMBL1140583 0.74 MEN1 (0.55) ALDH1A1POLBTDP1LMNASMN1; SMN2
SCHEMBL1140486 0.74 TDP1 (0.54) ALDH1A1POLBTDP1LMNAKDM4E
SCHEMBL1140535 0.74 ALDH1A1 (0.54) ALDH1A1POLBTDP1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230278971-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES VERSITECH LIMITED (HK) 2023-09-07 US disclosed
US-20230278971-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES VERSITECH LIMITED (HK) 2023-09-07 US disclosed
US-20210309622-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES VERSITECH LIMITED (HK) 2021-10-07 US disclosed
US-20210309622-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES VERSITECH LIMITED (HK) 2021-10-07 US disclosed
US-11052078-B2 Compounds affecting pigment production and methods for treatment of bacterial diseases VERSITECH LIMITED (CN) 2021-07-06 US disclosed
US-11052078-B2 Compounds affecting pigment production and methods for treatment of bacterial diseases VERSITECH LIMITED (CN) 2021-07-06 US disclosed
US-11040949-B2 Compounds affecting pigment production and methods for treatment of bacterial diseases VERSITECH LIMITED (CN) 2021-06-22 US disclosed
US-11040949-B2 Compounds affecting pigment production and methods for treatment of bacterial diseases VERSITECH LIMITED (CN) 2021-06-22 US disclosed
US-20200392095-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES THE UNIVERSITY OF HONG KONG (HK) 2020-12-17 US disclosed
US-20200392095-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES THE UNIVERSITY OF HONG KONG (HK) 2020-12-17 US disclosed
US-20200261438-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES THE UNIVERSITY OF HONG KONG (HK) 2020-08-20 US disclosed
US-20200261438-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES THE UNIVERSITY OF HONG KONG (HK) 2020-08-20 US disclosed
US-20190022038-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES VERSITECH LIMITED (HK) 2019-01-24 US disclosed
US-20190022038-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES VERSITECH LIMITED (HK) 2019-01-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11040949-B2 Compounds affecting pigment production and methods for treatment of bacterial diseases TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885
US-20200392095-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885
US-11052078-B2 Compounds affecting pigment production and methods for treatment of bacterial diseases TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885
US-20210309622-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885
US-20200261438-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885
US-20230278971-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885
US-20190022038-A1 COMPOUNDS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES TYR, ALAD, NQO1 ALDH1A1 295/4885POLB 212/4885RXFP1 4131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.