SCHEMBL206576

SCHEMBL206576

Cc1cnc(C(=O)N2CCN(C(=O)CCCC(=O)NC3CCC(Cc4ccccc4)(N(C)C)CC3)CC2)cn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
LMNA P02545 1/20 0.43
PRKAA2 P54646 4/20 0.40
PRKAB2 O43741 2/20 0.40
PRKAG1 P54619 2/20 0.40
PRKAA1 Q13131 2/20 0.40
PRKAG3 Q9UGI9 2/20 0.40
PRKAG2 Q9UGJ0 2/20 0.40
PRKAB1 Q9Y478 2/20 0.40
HTT P42858 1/20 0.39
OPRM1 P35372 2/20 0.38
OPRL1 P41146 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
C3AR1 Q16581 1/20 0.37
EPHX2 P34913 1/20 0.36
EPHX1 P07099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206152 0.88 POLB (0.37) ALDH1A1LMNAPRKAA2PRKAB2PRKAG1
SCHEMBL206115 0.87 NPC1 (0.38) ALDH1A1LMNAPRKAA2PRKAB2PRKAG1
SCHEMBL207964 0.86 ALDH1A1 (0.40) ALDH1A1LMNAPRKAA2PRKAB2PRKAG1
SCHEMBL205294 0.81 AR (0.56) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL206177 0.80 ALDH1A1 (0.48) ALDH1A1OPRM1OPRL1KMT2AEPHX2
SCHEMBL206079 0.80 OPRM1 (0.54) OPRM1OPRL1EPHX2EPHX1
SCHEMBL205791 0.79 MAPT (0.52) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL4072325 0.78 OPRM1 (0.52) LMNAOPRM1OPRL1EPHX2EPHX1
SCHEMBL207983 0.78 SIGMAR1 (0.50) ALDH1A1MEN1KMT2A
SCHEMBL206125 0.76 ADAMTS4 (0.47) ALDH1A1HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US claimed
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US disclosed