SCHEMBL2067900

SCHEMBL2067900

COc1ncccc1-c1nc2ccccc2c(N)c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.49
ACHE P22303 10/20 0.49
ADORA2A P29274 1/20 0.46
BCHE P06276 3/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 2/20 0.43
HPGD P15428 2/20 0.43
CASP1 P29466 2/20 0.43
CASP7 P55210 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CHRM1 P11229 1/20 0.43
NQO2 P16083 1/20 0.43
MAOA P21397 1/20 0.43
DRD1 P21728 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4821612 0.78 MAPT (0.51) DHODHMAPTKDM4EALDH1A1HPGD
SCHEMBL27952809 0.75 MTOR (0.48) ADORA2ABTKRAB9ANPC1
SCHEMBL2713912 0.73 S100A4 (0.49) BTKRAB9ANPC1
SCHEMBL8818671 0.72 TGFBR1 (0.49) DHODHMAPTALDH1A1LMNAPOLB
SCHEMBL13422264 0.71 DHODH (0.53) DHODHMAPTALDH1A1BTKRAB9A
SCHEMBL27944099 0.70 MTOR (0.49) ADORA2ABTKRAB9ANPC1
SCHEMBL18039110 0.70 MTOR (0.41) BTKRAB9ANPC1
SCHEMBL17492275 0.69 NPC1 (0.41) DHODHMAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL4056518 0.68 DHODH (0.54) DHODHMAPTALDH1A1CASP1BTK
SCHEMBL27915475 0.68 ADORA2A (0.51) ACHEADORA2ABCHEMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103030637-A Imidazole quinoline derivative, and pharmaceutically acceptable salts thereof, preparation method thereof and application thereof on medicines SHANGHAI HENGRUI PHARM CO LTD 2013-04-10 CN disclosed
EP-2438063-A1 1H-IMIDAZO[4,5-C]QUINOLINONE COMPOUNDS, USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES Novartis AG (CH) 2012-04-11 EP disclosed