SCHEMBL4821612

SCHEMBL4821612

COc1ncccc1-c1nc2ccccc2c(-c2ccncc2)c1-c1cccnc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.51
DHODH Q02127 1/20 0.47
KDM4E B2RXH2 4/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
PADI4 Q9UM07 1/20 0.42
SQOR Q9Y6N5 1/20 0.41
LMNA P02545 3/20 0.40
MAPK1 P28482 2/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 3/20 0.38
PDE10A Q9Y233 1/20 0.38
GAA P10253 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
USP2 O75604 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2067900 0.78 DHODH (0.49) MAPTDHODHKDM4EKMT2ALMNA
SCHEMBL29501236 0.73 BTK (0.50) MAPTDHODHSQORNPC1RAB9A
SCHEMBL13422264 0.70 DHODH (0.53) MAPTDHODHMEN1KMT2ASQOR
SCHEMBL29488279 0.69 ESR1 (0.58) MAPTDHODHKDM4EMEN1KMT2A
SCHEMBL9601498 0.69 ESR1 (0.58) MAPTDHODHKDM4EMEN1KMT2A
SCHEMBL1083765 0.68 MAPT (1.00) MAPTKDM4EMEN1KMT2ALMNA
SCHEMBL8818671 0.68 TGFBR1 (0.49) MAPTDHODHLMNAALDH1A1GAA
SCHEMBL4056518 0.67 DHODH (0.54) MAPTDHODHMEN1KMT2ASQOR
SCHEMBL21445639 0.65 MAPK14 (0.38) MAPTDHODHKDM4EMEN1KMT2A
SCHEMBL21445433 0.65 MAPK14 (0.38) MAPTDHODHKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008144463-A1 QUINOLINE DERIVATIVES AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-11-27 WO disclosed