SCHEMBL20733331

SCHEMBL20733331

COc1cc(C)cc(N(C)c2cccc(C)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.55
EGFR P00533 3/20 0.45
CSF1R P07333 3/20 0.45
MTNR1A P48039 6/20 0.44
MTNR1B P49286 6/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HSD17B1 P14061 6/20 0.41
HSD17B2 P37059 6/20 0.41
RELA Q04206 1/20 0.40
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2B P41595 1/20 0.38
CYP51A1 Q16850 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12012667 0.84 ACHE (0.52) ACHEEGFRCSF1RMTNR1AMTNR1B
SCHEMBL13367407 0.83 ACHE (0.55) ACHEEGFRCSF1RNPC1RAB9A
SCHEMBL1697445 0.81 ACHE (0.55) ACHEEGFRCSF1RNPC1RAB9A
SCHEMBL30054343 0.79 MTNR1A (0.61) ACHEMTNR1AMTNR1BHSD17B1HSD17B2
SCHEMBL1134082 0.79 MTNR1A (0.61) ACHEMTNR1AMTNR1BHSD17B1HSD17B2
SCHEMBL9853296 0.79 ACHE (0.53) ACHEEGFRCSF1RNPC1RAB9A
SCHEMBL10042868 0.77 MTNR1A (0.51) ACHEEGFRCSF1RMTNR1AMTNR1B
SCHEMBL22166438 0.77 MTNR1A (0.60) ACHEMTNR1AMTNR1BNPC1RAB9A
SCHEMBL10042849 0.77 ACHE (0.47) ACHEEGFRCSF1RMTNR1AMTNR1B
SCHEMBL8497577 0.77 ACHE (0.67) ACHEMTNR1AMTNR1BNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019032563-A1 INHIBITORS OF BASE EXCISION REPAIR ACTIVITY AND THERAPEUTIC METHODS BASED THEREON THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2019-02-14 WO disclosed