SCHEMBL2073780

SCHEMBL2073780

CCCCCCCCCC(CC(N)=O)(c1ccccc1)c1ncc[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 3/20 0.37
SCN9A Q15858 3/20 0.37
HSP90AA1 P07900 1/20 0.36
CYP3A4 P08684 2/20 0.34
OPRK1 P41145 2/20 0.34
MEN1 O00255 1/20 0.34
NR1I2 O75469 1/20 0.34
LMNA P02545 1/20 0.34
CHRM2 P08172 1/20 0.34
ADRA2A P08913 1/20 0.34
MAPT P10636 1/20 0.34
HTR2B P41595 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KIF11 P52732 1/20 0.33
SLC22A2 O15244 1/20 0.33
SLC22A1 O15245 1/20 0.33
PGR P06401 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2073778 0.81 CYP3A4 (0.43) SCN5ASCN9AHSP90AA1CYP3A4OPRK1
SCHEMBL15564307 0.78 SCN5A (0.40) SCN5ASCN9AHSP90AA1CYP3A4OPRK1
SCHEMBL2073783 0.76 MMP1 (0.37) SCN5ASCN9ACYP3A4OPRK1MEN1
SCHEMBL11804628 0.73 LMNA (0.36) HSP90AA1CYP3A4OPRK1LMNACHRM2
SCHEMBL11794861 0.72 CYP19A1 (0.35) HSP90AA1CYP3A4LMNAALOX15
SCHEMBL28833568 0.72 SCN5A (0.50) SCN5ASCN9ACYP3A4OPRK1MEN1
SCHEMBL11846314 0.71 TSHR (0.43) CYP3A4MEN1LMNACHRM2KMT2A
SCHEMBL8978824 0.69 ESR1 (0.53) SCN5ASCN9AMEN1KMT2AGAA
SCHEMBL4740369 0.69 ESR1 (0.53) SCN5ASCN9AMEN1KMT2AGAA
SCHEMBL10448023 0.69 ESR1 (0.53) SCN5ASCN9AMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863294-B2 Heterocycle derivatives as histone deacetylase (HDAC) inhibitors INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-01-04 US disclosed