SCHEMBL2073778

SCHEMBL2073778

CCCCCCCCCCC(C(N)=O)(c1ccccc1)c1ncc[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.43
KCNH2 Q12809 2/20 0.43
OPRK1 P41145 2/20 0.43
TSHR P16473 2/20 0.43
BLM P54132 2/20 0.43
PMP22 Q01453 2/20 0.43
SLC22A2 O15244 1/20 0.43
SLC22A1 O15245 1/20 0.43
PGR P06401 1/20 0.43
THRB P10828 1/20 0.43
ADRB3 P13945 1/20 0.43
PDE3A Q14432 1/20 0.43
SLC47A1 Q96FL8 1/20 0.43
ALOX15 P16050 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SCN5A Q14524 3/20 0.41
SCN9A Q15858 3/20 0.41
OPRM1 P35372 2/20 0.39
DRD3 P35462 2/20 0.39
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18248486 0.82 CHRM3 (0.54) CYP3A4KCNH2OPRK1TSHRBLM
SCHEMBL7643094 0.82 CHRM3 (0.54) CYP3A4KCNH2OPRK1TSHRBLM
SCHEMBL18248596 0.82 CHRM3 (0.54) CYP3A4KCNH2OPRK1TSHRBLM
SCHEMBL2073780 0.81 SCN5A (0.37) CYP3A4KCNH2OPRK1TSHRBLM
SCHEMBL2073783 0.80 MMP1 (0.37) CYP3A4OPRK1SCN5ASCN9ACHRM2
SCHEMBL15564302 0.77 SCN5A (0.44) CYP3A4KCNH2OPRK1TSHRBLM
SCHEMBL15564219 0.77 SCN5A (0.44) CYP3A4KCNH2OPRK1TSHRBLM
Phosphoric Acid SCHEMBL3688742 0.77 CHRM2 (0.49) KCNH2SCN5ASCN9AOPRM1DRD3
Phosphoric Acid SCHEMBL29728497 0.77 CHRM2 (0.49) KCNH2SCN5ASCN9AOPRM1DRD3
SCHEMBL2984162 0.76 CHRM3 (0.56) CYP3A4KCNH2OPRK1TSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863294-B2 Heterocycle derivatives as histone deacetylase (HDAC) inhibitors INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-01-04 US disclosed