SCHEMBL20788239

SCHEMBL20788239

Cc1cc(C(N)=O)nn1-c1ccc(Cc2ccc(Cl)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.56
SCN9A Q15858 7/20 0.51
NPY5R Q15761 1/20 0.46
MALT1 Q9UDY8 6/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
PPP1CA P62136 1/20 0.44
RPA1 P27694 1/20 0.43
CHRNA7 P36544 1/20 0.43
PTGER1 P34995 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15167854 0.92 L3MBTL1 (0.64) L3MBTL1SCN9ANPY5RMALT1NFKB1
SCHEMBL20788373 0.88 SMN1; SMN2 (0.57) L3MBTL1NPY5RMALT1NFKB1NFKB2
SCHEMBL20788274 0.85 SCN9A (0.55) SCN9ANPY5RHPGD
SCHEMBL20788268 0.84 CYP17A1 (0.50) L3MBTL1SCN9A
SCHEMBL20788403 0.84 CHRNA7 (0.56) TP53HPGDCHRNA7
SCHEMBL20788407 0.83 L3MBTL1 (0.54) L3MBTL1SCN9ANPY5RMALT1SMN1; SMN2
SCHEMBL20788386 0.83 SCN9A (0.45) L3MBTL1SCN9A
SCHEMBL20788432 0.83 SCN9A (0.45) L3MBTL1SCN9ATP53HPGDSMN1; SMN2
SCHEMBL20788211 0.81 HRH3 (0.47) L3MBTL1SCN9A
SCHEMBL20788440 0.81 HRH3 (0.44) L3MBTL1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3681883-B1 DIPHENYL DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2024-02-21 EP disclosed
CN-111094278-B Diphenyl derivative and use thereof 诺华股份有限公司 2023-07-14 CN disclosed
EP-3681883-A1 DIPHENYL DERIVATIVES AND USES THEREOF Novartis AG (CH) 2020-07-22 EP disclosed
CN-111094278-A Diphenyl derivatives and their use 诺华股份有限公司 2020-05-01 CN disclosed
US-10633350-B2 Diphenyl derivatives and uses thereof NOVARTIS AG (CH) 2020-04-28 US disclosed
US-10633350-B2 Diphenyl derivatives and uses thereof NOVARTIS AG (CH) 2020-04-28 US disclosed
WO-2019053090-A1 DIPHENYL DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2019-03-21 WO disclosed
US-20190077773-A1 DIPHENYL DERIVATIVES AND USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2019-03-14 US disclosed
US-20190077773-A1 DIPHENYL DERIVATIVES AND USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2019-03-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190077773-A1 DIPHENYL DERIVATIVES AND USES THEREOF MYOF, NGF, MUSK L3MBTL1 1366/4885SCN9A 2916/4885NPY5R 3243/4885
US-10633350-B2 Diphenyl derivatives and uses thereof MYOF, NGF, MUSK L3MBTL1 1366/4885SCN9A 2916/4885NPY5R 3243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.