SCHEMBL20837136

SCHEMBL20837136

Nc1[nH]nc(C(F)(F)F)c1-c1cc(F)cc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.37
NOTUM Q6P988 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SGK1 O00141 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20837143 0.84 IKBKB (0.43) IKBKBNOTUML3MBTL1MEN1KMT2A
SCHEMBL20837397 0.83 MAPK14 (0.43) NOTUML3MBTL1MEN1KMT2A
SCHEMBL2235270 0.83 IKBKB (0.37) IKBKBNOTUML3MBTL1SGK1
SCHEMBL20837302 0.78 ENPP1 (0.41) IKBKBL3MBTL1MEN1KMT2A
SCHEMBL1279682 0.75 IKBKB (0.46) IKBKBL3MBTL1SGK1MEN1KMT2A
SCHEMBL1846643 0.74 IKBKB (0.50) IKBKBNOTUML3MBTL1
SCHEMBL20837303 0.73 ENPP1 (0.48) IKBKBNOTUML3MBTL1MEN1KMT2A
SCHEMBL20837280 0.72 GAA (0.36) IKBKBL3MBTL1SGK1MEN1KMT2A
SCHEMBL20837142 0.72 MAPT (0.46) MEN1KMT2A
SCHEMBL20837311 0.71 KIF11 (0.45) NOTUML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10738056-B2 Pyrazolopyrimidinone compounds and uses thereof ADURO BIOTECH INC. (US) 2020-08-11 US disclosed
US-20190119285-A1 PYRAZOLOPYRIMIDINONE COMPOUNDS AND USES THEREOF CHINOOK THERAPEUTICS, INC. 2019-04-25 US disclosed
WO-2019055750-A1 PYRAZOLOPYRIMIDINONE COMPOUNDS AND USES THEREOF Aduro Biotech, Inc. (US) 2019-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10738056-B2 Pyrazolopyrimidinone compounds and uses thereof NLRP3, NLRP1, P2RX7 IKBKB 1662/4885NOTUM 423/4885L3MBTL1 4818/4885
US-20190119285-A1 PYRAZOLOPYRIMIDINONE COMPOUNDS AND USES THEREOF NLRP3, NLRP1, P2RX7 IKBKB 1662/4885NOTUM 423/4885L3MBTL1 4818/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.