SCHEMBL20846009

SCHEMBL20846009

CC(=O)N(C)c1ncc(-c2cncc(F)c2)nc1C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.37
CYP11B2 P19099 7/20 0.35
PIK3CG P48736 1/20 0.35
CYP11B1 P15538 2/20 0.34
ABL1 P00519 4/20 0.33
HCAR2 Q8TDS4 1/20 0.33
GRM1 Q13255 1/20 0.32
PARP10 Q53GL7 1/20 0.32
PARP11 Q9NR21 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
GRIN2B Q13224 2/20 0.32
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839273 0.88 CYP11B2 (0.38) PIM1CYP11B2PIK3CGCYP11B1ABL1
SCHEMBL29911053 0.84 PIM1 (0.42) PIM1CYP11B2CYP11B1PARP10PARP11
SCHEMBL20839010 0.84 PIM1 (0.42) PIM1CYP11B2CYP11B1PARP10PARP11
SCHEMBL20839344 0.83 TLR7 (0.34) PIM1ABL1HCRTR1HCRTR2
SCHEMBL24013138 0.83 PIM1 (0.34) PIM1CYP11B2PIK3CGCYP11B1ABL1
SCHEMBL20843700 0.80 TLR7 (0.40) ABL1
SCHEMBL20839266 0.77 TLR7 (0.34) PIM1CYP11B2ABL1HCRTR1HCRTR2
SCHEMBL20846011 0.75 PIK3CG (0.46) PIM1CYP11B2PIK3CGCYP11B1ABL1
SCHEMBL20839264 0.75 CYP11B2 (0.36) PIM1CYP11B2PIK3CGCYP11B1ABL1
SCHEMBL20839015 0.72 PIM1 (0.43) PIM1CYP11B2CYP11B1PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11678665-B2 Pyrazine-4-carbamate or -urea derivatives as herbicides SYNGENTA PARTICIPATIONS AG (CH) 2023-06-20 US disclosed
US-11678665-B2 Pyrazine-4-carbamate or -urea derivatives as herbicides SYNGENTA PARTICIPATIONS AG (CH) 2023-06-20 US disclosed
EP-3684764-B1 PYRAZINE-4-CARBAMATE DERIVATIVES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2021-11-10 EP disclosed
US-20200267983-A1 Pyrazine-4Carbamate or -Urea Derivatives As Herbicides SYNGENTA PARTICIPATIONS AG (CH) 2020-08-27 US disclosed
WO-2019057724-A1 PYRAZINE-4CARBAMATE OR -UREA DERIVATIVES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2019-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11678665-B2 Pyrazine-4-carbamate or -urea derivatives as herbicides DDT, PLPBP, CPS1 PIM1 1335/4885CYP11B2 3239/4885PIK3CG 926/4885
US-20200267983-A1 Pyrazine-4Carbamate or -Urea Derivatives As Herbicides PLPBP, PDXK, HPD PIM1 1700/4885CYP11B2 3269/4885PIK3CG 874/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.