SCHEMBL20856347

SCHEMBL20856347

O=[N+]([O-])c1cc(CC(F)(F)F)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
VCAM1 P19320 14/20 0.47
TDP1 Q9NUW8 2/20 0.46
KDM1A O60341 1/20 0.44
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
HIF1A Q16665 1/20 0.42
TXNRD1 Q16881 1/20 0.42
TXNRD3 Q86VQ6 1/20 0.42
TXNRD2 Q9NNW7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28771294 0.87 TSHR (0.53) ALDH1A1VCAM1TDP1CYP3A4HPGD
SCHEMBL28179842 0.84 TSHR (0.46) ALDH1A1POLBTDP1CYP3A4HPGD
SCHEMBL9913587 0.81 ALDH1A1 (0.53) ALDH1A1VCAM1TDP1HIF1A
SCHEMBL31023123 0.81 ALDH1A1 (0.53) ALDH1A1VCAM1TDP1HIF1A
SCHEMBL27311122 0.81 VCAM1 (0.51) ALDH1A1KDM4EPOLBVCAM1TDP1
SCHEMBL27555022 0.80 ALDH1A1 (0.43) ALDH1A1KDM4EPOLBTDP1CYP3A4
SCHEMBL8790573 0.80 TDP1 (0.58) ALDH1A1POLBTDP1CYP3A4ALOX15
SCHEMBL27565845 0.80 PARP1 (0.45) ALDH1A1POLBTDP1CYP3A4HPGD
SCHEMBL4520586 0.79 VCAM1 (0.53) ALDH1A1KDM4EPOLBVCAM1TDP1
SCHEMBL27304953 0.79 ALDH1A1 (0.41) ALDH1A1KDM4EPOLBVCAM1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103274945-A Cleaning and preparing method of 4-Chloro-3,5-dinitrobenzotrifluoride JIANGSU DAHUA CHEMICAL IND CO LTD 2013-09-04 CN claimed
CN-103265435-A Clean preparation method of 4-chlorine-3-nitrobenzotrifluoride JIANGSU DAHUA CHEMICAL IND CO LTD 2013-08-28 CN claimed
CN-103102284-A Preparation of 4-trifluoromethyl-2, 6-dinitrobenzene salicylaldoxime derivative and its application in anticancer therapeutic drugs NANJING UNIVERSITY OF TECHNOLOGY 2013-05-15 CN claimed
US-20210147408-A1 SMALL MOLECULE INHIBITORS OF GALECTIN-3 BRISTOL MYERS SQUIBB CO (US) 2021-05-20 US disclosed
US-20210147408-A1 SMALL MOLECULE INHIBITORS OF GALECTIN-3 BRISTOL MYERS SQUIBB CO (US) 2021-05-20 US disclosed
CN-109320396-B Preparation method of octafluorotoluene 湖南有色郴州氟化学有限公司 2021-03-19 CN disclosed
WO-2019067702-A9 SMALL MOLECULE INHIBITORS OF GALECTIN-3 BRISTOL-MYERS SQUIBB COMPANY (US) 2019-04-25 WO disclosed
WO-2019067702-A1 SMALL MOLECULE INHIBITORS OF GALECTIN-3 BRISTOL-MYERS SQUIBB COMPANY (US) 2019-04-04 WO disclosed
CN-103755572-B A kind of trifluralin nitrated workshop section spent acid circulation use technology JIANGSU FENGSHAN GROUP CO., LTD. (CN) 2016-03-02 CN disclosed
CN-104926691-A Preparation method of 2-nitro-4-trifluoromethylbenzonitrile JIANGSU AGROCHEM LAB CO LTD 2015-09-23 CN disclosed
CN-103274945-A Cleaning and preparing method of 4-Chloro-3,5-dinitrobenzotrifluoride JIANGSU DAHUA CHEMICAL IND CO LTD 2013-09-04 CN disclosed
CN-1051313-C 5-arylindole derivatives PFIZER (US) 2000-04-12 CN disclosed
CN-1038749-C Dibenz [b,f] [1,4] oxazepin-11(10H)-ones for multidrug resistance reversing agents BRISTOL MYERS SQUIBB CO (US) 1998-06-17 CN disclosed
CN-1161334-A Novel substd. guanidine derivs., process for prodn. thereof, and pharmaceutical uses thereof SUMITOMO PHARMA (JP) 1997-10-08 CN disclosed
CN-1152918-A Novel amido quinoxaline diones, their preparation and use BASF AG (DE) 1997-06-25 CN disclosed
CN-1094727-A The 5-(hetero) aryl indole derivatives PFIZER (US) 1994-11-09 CN disclosed
CN-1025855-C Process and intermediates for prepation of oxophthalazinyl acetic acids and analogs thereof PFIZER (US) 1994-09-07 CN disclosed
CN-1072679-A INDOLE DERIVATIVES PFIZER (US) 1993-06-02 CN disclosed
CN-1069731-A Dibenzo [b, f] [1,4] oxygen azepine -11 (10H) ketone that is used for multiple drug resistance reversal agent BRISTOL MYERS SQUIBB CO (US) 1993-03-10 CN disclosed
CN-1047499-A The method and the intermediate that prepare oxo phthalazinyl acetate and homologue PFIZER (US) 1990-12-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210147408-A1 SMALL MOLECULE INHIBITORS OF GALECTIN-3 LGALS3, LGALS1, LGALS3BP ALDH1A1 2893/4885KDM4E 3932/4885POLB 4830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.