SCHEMBL20877908

SCHEMBL20877908

CCOC(=O)/C(=N\NC(=O)OC(C)(C)C)C(=O)COCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.43
SYK P43405 1/20 0.43
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NPC1 O15118 3/20 0.42
AKT1 P31749 3/20 0.41
ALDH1A1 P00352 1/20 0.41
CTSS P25774 3/20 0.41
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
PPARG P37231 1/20 0.39
CTSL P07711 2/20 0.38
CTSB P07858 2/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CSNK1D P48730 1/20 0.38
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16559310 1.00 PPARA (0.43) PPARASYKRAB9ASMN1; SMN2NPC1
SCHEMBL6852186 0.81 NPC1 (0.51) PPARASYKRAB9ASMN1; SMN2NPC1
SCHEMBL21201525 0.79 ATM (0.44) RAB9ASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL16561964 0.78 CTSK (0.36) ALDH1A1KMT2A
SCHEMBL16577823 0.78 CTSK (0.36) ALDH1A1KMT2A
SCHEMBL16578523 0.78 GAA (0.41) RAB9ASMN1; SMN2NPC1ALDH1A1MEN1
SCHEMBL20877907 0.78 ALDH1A1 (0.42) RAB9ASMN1; SMN2NPC1ALDH1A1MEN1
SCHEMBL16559321 0.78 ALDH1A1 (0.42) RAB9ASMN1; SMN2NPC1ALDH1A1MEN1
SCHEMBL22704140 0.77 NPC1 (0.40) PPARARAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL25037571 0.77 MAPT (0.39) RAB9ASMN1; SMN2NPC1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210186969-A1 AZA-PYRIDONE COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-06-24 US disclosed
US-10980805-B2 Aza-pyridone compounds and uses thereof Janssen Biopharma, Inc. (US) 2021-04-20 US disclosed
US-20200030328-A1 AZA-PYRIDONE COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2020-01-30 US disclosed
US-10251882-B2 Aza-pyridone compounds and uses thereof ALIOS BIOPHARMA, INC. (US) 2019-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200030328-A1 AZA-PYRIDONE COMPOUNDS AND USES THEREOF PNPO, ITPA, PDXK PPARA 1459/4885SYK 3092/4885RAB9A 1824/4885
US-10980805-B2 Aza-pyridone compounds and uses thereof PNPO, ITPA, PDXK PPARA 1459/4885SYK 3092/4885RAB9A 1824/4885
US-10251882-B2 Aza-pyridone compounds and uses thereof PNPO, ITPA, PDXK PPARA 1459/4885SYK 3092/4885RAB9A 1824/4885
US-20210186969-A1 AZA-PYRIDONE COMPOUNDS AND USES THEREOF PNPO, ITPA, PDXK PPARA 1459/4885SYK 3092/4885RAB9A 1824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.