SCHEMBL20880131

SCHEMBL20880131

CNCc1ccc(C(=N)CN)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.44
NOS3 P29474 1/20 0.44
NOS2 P35228 1/20 0.44
LOXL2 Q9Y4K0 3/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
F10 P00742 1/20 0.39
CA2 P00918 1/20 0.38
NCF1 P14598 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
PTGS2 P35354 1/20 0.37
PLK1 P53350 1/20 0.36
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL48986 0.80 PRSS1 (0.57) NOS1NOS3NOS2LOXL2F10
SCHEMBL20880151 0.77 LOXL2 (0.64) NOS1NOS3NOS2LOXL2F10
SCHEMBL2504209 0.73 KDM4E (0.68) NOS1NOS3NOS2LOXL2KDM4E
SCHEMBL25910898 0.73 ALDH1A1 (0.42) LOXL2F10ALDH1A1LMNACYP1A2
SCHEMBL22872694 0.72 NOS1 (0.52) NOS1NOS3NOS2LOXL2KDM4E
SCHEMBL16181585 0.72 NOS1 (0.52) NOS1NOS3NOS2LOXL2KDM4E
SCHEMBL3882642 0.72 PLA2G10 (0.57) NOS1NOS3NOS2LOXL2KDM4E
SCHEMBL4865180 0.72 KDM4E (0.54) NOS1NOS3NOS2LOXL2KDM4E
Hydrochloric Acid SCHEMBL30925271 0.71 KDM4E (0.74) NOS1NOS3NOS2LOXL2KDM4E
Hydrochloric Acid SCHEMBL10921172 0.70 KDM4E (0.44) NOS1NOS3NOS2LOXL2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3466961-A1 PROLINAMIDE DERIVATIVE AS THROMBIN INHIBITOR, PREPARATION METHOD AND APPLICATION THEREOF Li, Min (US) 2019-04-10 EP disclosed