SCHEMBL2089394

SCHEMBL2089394

COC(=O)Nc1ccc(OC)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.73
NPC1 O15118 6/20 0.73
RAB9A P51151 6/20 0.73
HPGD P15428 2/20 0.70
CYP1A2 P05177 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
TP53 P04637 2/20 0.66
ALOX15 P16050 1/20 0.66
ALDH1A1 P00352 2/20 0.65
HTT P42858 2/20 0.65
GAA P10253 1/20 0.65
TGM2 P21980 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
MAPT P10636 3/20 0.59
KDM4E B2RXH2 1/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
SAE1 Q9UBE0 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9609808 0.89 SMN1; SMN2 (0.82) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL11773292 0.87 SMN1; SMN2 (0.85) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL2089392 0.86 RAB9A (0.66) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL11092496 0.84 RAB9A (1.00) SMN1; SMN2NPC1RAB9ATP53ALOX15
SCHEMBL6396790 0.84 RAB9A (0.76) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL1342005 0.83 SMN1; SMN2 (0.61) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL9357891 0.83 RAB9A (1.00) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL7556396 0.83 NPC1 (0.69) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL992202 0.83 RAB9A (0.73) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL171415 0.83 SMN1; SMN2 (0.73) SMN1; SMN2NPC1RAB9ACYP1A2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081481-B2 Excitatory amino acid receptor modulators ELI LILLY AND COMPANY (US) 2006-07-25 US claimed
US-20040102521-A1 Excitatory amino acid receptor modulators ELI LILLY AND COMPANY 2004-05-27 US claimed
EP-1289940-A2 EXCITATORY AMINO ACID RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2003-03-12 EP claimed
WO-2001092213-A2 EXCITATORY AMINO ACID RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2001-12-06 WO claimed
US-5091556-A Catalytic reacting carbonate with amine ENICHEM SYNTHESIS, S.P.A. (IT) 1992-02-25 US claimed
CN-122011028-A Method for efficiently preparing various substituted chiral phosphoramides 上海交通大学 2026-05-12 CN disclosed
CN-113474347-A AZA heterobicyclic inhibitors of MAT2A and methods for treating cancer 法国施维雅药厂 2021-10-01 CN disclosed
EP-3508473-B1 METHOD FOR PRODUCING CARBAMIC ACID ESTER AIST (JP) 2021-05-26 EP disclosed
WO-2020251953-A1 STREPTOGRAMIN COMPOSITIONS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-12-17 WO disclosed
US-10752579-B2 Production method of carbamic acid ester NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 2020-08-25 US disclosed
EP-3508473-A1 METHOD FOR PRODUCING CARBAMIC ACID ESTER National Institute of Advanced Industrial Science and Technology (JP) 2019-07-10 EP disclosed
US-20190185420-A1 PRODUCTION METHOD OF CARBAMIC ACID ESTER NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 2019-06-20 US disclosed
US-20040102521-A1 Excitatory amino acid receptor modulators ELI LILLY AND COMPANY 2004-05-27 US disclosed
EP-1289940-A2 EXCITATORY AMINO ACID RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
CN-1331688-A Aminopyridine Derivatives TEIKOKU HORMONE MFG CO LTD (JP) 2002-01-16 CN disclosed
WO-2001092213-A2 EXCITATORY AMINO ACID RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2001-12-06 WO disclosed
EP-0391473-B1 Process for producing carbamates ENICHEM SINTESI (IT) 1994-05-04 EP disclosed
US-5091556-A Catalytic reacting carbonate with amine ENICHEM SYNTHESIS, S.P.A. (IT) 1992-02-25 US disclosed
EP-0391473-A1 Process for producing carbamates ENICHEM SYNTHESIS S.p.A. (IT) 1990-10-10 EP disclosed
US-4600797-A NITRATING AN AMINOBENZENE WHICH HAS A PROTECTEDD AMINO GROUP BAYER AKTIENGESELLSCHAFT (DE) 1986-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040102521-A1 Excitatory amino acid receptor modulators GRM1, GRM2, GRIN1 SMN1; SMN2 1182/4885NPC1 1241/4885RAB9A 2180/4885
US-20190185420-A1 PRODUCTION METHOD OF CARBAMIC ACID ESTER CA2, CA7, CA4 SMN1; SMN2 3068/4885NPC1 2799/4885RAB9A 2467/4885
US-10752579-B2 Production method of carbamic acid ester CA2, CA7, CA4 SMN1; SMN2 3068/4885NPC1 2799/4885RAB9A 2467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.