SCHEMBL20894366

SCHEMBL20894366

COCCNc1ccc(B2OC(C)(C)C(C)(C)O2)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.50
DGAT1 O75907 3/20 0.47
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
USP30 Q70CQ3 1/20 0.38
LPL P06858 4/20 0.38
LIPG Q9Y5X9 4/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
MKNK1 Q9BUB5 2/20 0.37
FYN P06241 2/20 0.37
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 3/20 0.35
ALOX15 P16050 2/20 0.35
HSD17B10 Q99714 2/20 0.35
HIF1A Q16665 1/20 0.35
USP2 O75604 1/20 0.35
APEX1 P27695 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29630971 1.00 HCAR3 (0.50) HCAR3DGAT1ALDH1A1KDM4EUSP30
SCHEMBL2601997 0.92 DGAT1 (0.46) HCAR3DGAT1ALDH1A1KDM4EUSP30
SCHEMBL25066062 0.83 DGAT1 (0.46) HCAR3DGAT1USP30LPLLIPG
SCHEMBL182973 0.83 DGAT1 (0.46) HCAR3DGAT1ALDH1A1KDM4EUSP30
SCHEMBL22674352 0.83 DGAT1 (0.43) DGAT1USP30LPLLIPGCA1
SCHEMBL19996746 0.83 DGAT1 (0.43) DGAT1USP30LPLLIPGCA1
SCHEMBL1842384 0.83 DGAT1 (0.41) HCAR3DGAT1ALDH1A1KDM4EUSP30
SCHEMBL25698622 0.81 LRRK2 (0.43) HCAR3DGAT1ALDH1A1KDM4ECYP1A2
SCHEMBL2432651 0.81 LPL (0.50) HCAR3DGAT1LPLLIPGCA1
SCHEMBL31262570 0.81 CYP2C19 (0.47) DGAT1USP30LPLLIPGMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340551-A1 SMALL MOLECULE MODULATORS OF STAT6 GILEAD SCIENCES INC (US) 2025-11-06 US disclosed
US-20250325677-A1 STAT6 DEGRADERS GILEAD SCIENCES INC (US) 2025-10-23 US disclosed
US-20220213103-A1 9H-PYRROLO-DIPYRIDINE DERIVATIVES UCB Biopharma SRL (BE) 2022-07-07 US disclosed
CN-109563094-B (hetero) aryl-substituted piperidinyl derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2022-03-18 CN disclosed
US-10654849-B2 (Hetero)aryl-substituted-piperidinyl derivatives, a process for their preparation and pharmaceutical compositions containing them LES LABORATOIRES SERVIER (FR) 2020-05-19 US disclosed
EP-3468971-B1 NEW (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2020-02-19 EP disclosed
US-20190144449-A1 (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2019-05-16 US disclosed
EP-3468971-A1 NEW (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Les Laboratoires Servier (FR) 2019-04-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220213103-A1 9H-PYRROLO-DIPYRIDINE DERIVATIVES MAPT, PSEN1, PRNP HCAR3 3079/4885DGAT1 4778/4885ALDH1A1 3567/4885
US-20250325677-A1 STAT6 DEGRADERS STAT6, STAT5B, STAT1 HCAR3 721/4885DGAT1 1054/4885ALDH1A1 959/4885
US-20250340551-A1 SMALL MOLECULE MODULATORS OF STAT6 STAT6, STAT1, STAT5B HCAR3 1332/4885DGAT1 661/4885ALDH1A1 2050/4885
US-20190144449-A1 (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BAX, BCL2, CCNK HCAR3 3194/4885DGAT1 4420/4885ALDH1A1 1524/4885
US-10654849-B2 (Hetero)aryl-substituted-piperidinyl derivatives, a process for their preparation and pharmaceutical compositions containing them BAX, BCL2, CCNK HCAR3 3194/4885DGAT1 4420/4885ALDH1A1 1524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.