SCHEMBL20938540

SCHEMBL20938540

C=C(S/C(C)=N\C)c1ccc2cnc(NC(=C)N3CCC(NC)CC3)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 18/20 0.43
GSK3B P49841 15/20 0.43
WNT1 P04628 4/20 0.39
CCNK O75909 2/20 0.35
CCNA2 P20248 2/20 0.35
CDK2 P24941 2/20 0.35
CDK7 P50613 2/20 0.35
CCNH P51946 2/20 0.35
MNAT1 P51948 2/20 0.35
CDK12 Q9NYV4 2/20 0.35
CLK2 P49760 1/20 0.33
CLK3 P49761 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20938647 0.80 DYRK1A (0.45) DYRK1AGSK3BWNT1
SCHEMBL20938744 0.79 DYRK1A (0.46) DYRK1AGSK3BWNT1CCNKCCNA2
SCHEMBL19546936 0.79 HCAR3 (0.33) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL20938656 0.79 DYRK1A (0.50) DYRK1AGSK3BWNT1CCNKCCNA2
SCHEMBL24219615 0.77 GSK3B (0.37) DYRK1AGSK3BWNT1
SCHEMBL23741124 0.76 GSK3B (0.51) DYRK1AGSK3BWNT1CCNKCCNA2
SCHEMBL23740951 0.75 GSK3B (0.59) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL23740979 0.75 GSK3B (0.58) DYRK1AGSK3BWNT1
SCHEMBL23741126 0.74 DYRK1A (0.56) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL23740875 0.73 DYRK1A (0.32) DYRK1AGSK3BWNT1CLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019079626-A1 6-(5-MEMBERED HETEROARYL)ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF SAMUMED, LLC (US) 2019-04-25 WO disclosed