SCHEMBL2097005

SCHEMBL2097005

Nc1nc(N)c(N)c(OCc2ccc(CNC(=O)C(F)(F)F)cc2)n1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.67
MGMT P16455 9/20 0.45
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
MPO P05164 4/20 0.41
DHFR P00374 2/20 0.36
GHSR Q92847 1/20 0.36
TPO P07202 1/20 0.35
CYP3A4 P08684 1/20 0.35
EPX P11678 1/20 0.35
CDK5 Q00535 1/20 0.35
TAOK1 Q7L7X3 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2100316 0.87 MGMT (0.63) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL2775958 0.81 PIN1 (0.73) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL3425790 0.80 PIN1 (1.00) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL29795745 0.80 PIN1 (1.00) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL2096999 0.80 MGMT (0.44) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL2098363 0.79 PIN1 (0.58) PIN1MGMTCDK2MPOCDK5
SCHEMBL2097456 0.78 PIN1 (0.62) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL2097362 0.78 PIN1 (0.62) PIN1MGMTMPODHFRTPO
SCHEMBL2748645 0.78 PIN1 (0.57) PIN1CDK2CDK5TAOK1CLK4
SCHEMBL2747687 0.77 PIN1 (0.56) PIN1CDK2MPOCDK5TAOK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730298-B1 SPECIFIC SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE EPFL ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (CH) 2015-11-11 EP disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase EPFL ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase AGT, AGXT, AGTR1 PIN1 2756/4885MGMT 303/4885CDK1 833/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.