SCHEMBL2097346

SCHEMBL2097346

CC(C)(C)OC(=O)NCCCC(=O)Nc1nc(N)nc(OCc2ccc(CNC(=O)C(F)(F)F)cc2)c1N=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.47
CA1 P00915 5/20 0.45
CA2 P00918 5/20 0.45
HDAC1 Q13547 1/20 0.39
CYP3A4 P08684 1/20 0.38
MGMT P16455 3/20 0.38
TLR7 Q9NYK1 3/20 0.37
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
KDM4E B2RXH2 2/20 0.34
POLB P06746 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
PAX8 Q06710 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14383622 0.88 CDK1 (0.47) CA1CA2HDAC1CYP3A4MGMT
SCHEMBL14383623 0.84 HDAC8 (0.41) CA1CA2HDAC1CYP3A4MGMT
SCHEMBL2056437 0.82 CA1 (0.43) CA1CA2CYP3A4TLR7L3MBTL1
SCHEMBL17244386 0.80 PIN1 (0.49) PIN1CA1CA2HDAC1CYP3A4
SCHEMBL2100316 0.76 MGMT (0.63) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL2054842 0.76 PIN1 (0.51) PIN1CA1CA2HDAC1L3MBTL1
SCHEMBL2099420 0.76 PIN1 (0.52) PIN1CA1CA2HDAC1CYP3A4
SCHEMBL14383628 0.71 PIN1 (0.51) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL2097005 0.69 PIN1 (0.67) PIN1CYP3A4MGMTCDK1CCNB1
SCHEMBL23148223 0.69 L3MBTL1 (0.55) CA1CA2HDAC1L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730298-B1 SPECIFIC SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE EPFL ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (CH) 2015-11-11 EP disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase EPFL ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase AGT, AGXT, AGTR1 PIN1 2756/4885CA1 4500/4885CA2 3221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.