SCHEMBL2097438

SCHEMBL2097438

Nc1nc2c(ncn2-c2cc(Br)cs2)c(=O)[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 9/20 0.55
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
PNP P00491 3/20 0.44
TK1 P04183 2/20 0.43
BLM P54132 2/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
EDNRA P25101 1/20 0.43
HTR2A P28223 1/20 0.43
RECQL P46063 1/20 0.43
HBB P68871 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
NFKB1 P19838 1/20 0.41
VCP P55072 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1899765 0.78 XDH (0.64) XDHMEN1KMT2APNPTK1
SCHEMBL3310025 0.77 XDH (0.76) XDHMEN1KMT2APNPTK1
SCHEMBL21629986 0.77 PNP (0.58) MEN1KMT2APNPTK1BLM
SCHEMBL1286945 0.71 XDH (1.00) XDHMEN1KMT2APNPTK1
SCHEMBL28095386 0.71 XDH (0.57) XDHMEN1KMT2APNPTK1
SCHEMBL986800 0.71 XDH (0.60) XDHMEN1KMT2APNPTK1
Hydrochloric Acid SCHEMBL21799342 0.70 XDH (0.97) XDHMEN1KMT2APNPTK1
SCHEMBL21417341 0.70 XDH (0.53) XDHMEN1KMT2APNPTK1
SCHEMBL41787 0.70 XDH (0.59) XDHMEN1KMT2APNPTK1
SCHEMBL15005119 0.70 XDH (0.59) XDHMEN1KMT2APNPTK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730298-B1 SPECIFIC SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE EPFL ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (CH) 2015-11-11 EP disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed