SCHEMBL210190

SCHEMBL210190

O=C(O)c1ccc(Nc2nccc(-c3cccnc3)n2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 10/20 0.76
BCR P11274 9/20 0.76
PRKCA P17252 5/20 0.76
PRKCD Q05655 4/20 0.75
EGFR P00533 1/20 0.75
CAMK2D Q13557 3/20 0.74
MAPK8 P45983 2/20 0.67
MAPK10 P53779 1/20 0.67
HDAC1 Q13547 1/20 0.65
GSK3B P49841 2/20 0.65
PIK3CG P48736 1/20 0.65
CAMKK2 Q96RR4 1/20 0.65
SRC P12931 5/20 0.63
PDGFRB P09619 4/20 0.63
PDGFRA P16234 4/20 0.63
PRKD3 O94806 1/20 0.63
PRKCG P05129 1/20 0.63
PRKCB P05771 1/20 0.63
PRKCH P24723 1/20 0.63
PRKCI P41743 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7470853 0.99 ABL1 (0.74) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL7467179 0.88 ABL1 (0.69) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL4903328 0.88 MAPK8 (0.81) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL7470849 0.88 ABL1 (0.69) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL7464657 0.86 CAMK2D (0.90) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL1655099 0.86 ABL1 (1.00) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL7474316 0.86 HDAC1 (0.68) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL6262145 0.86 ABL1 (1.00) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL4903275 0.85 ABL1 (0.81) ABL1BCRPRKCAPRKCDEGFR
SCHEMBL7464205 0.85 ABL1 (0.76) ABL1BCRPRKCAPRKCDEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922309-B1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF IL YANG PHARM CO LTD (KR) 2014-05-21 EP disclosed
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-7501424-B2 N-phenyl-2-pyrimidine-amine derivatives and process for the preparation thereof IL-YANG PHARM. CO., LTD. (KR) 2009-03-10 US disclosed
EP-1922309-A1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Il Yang Pharm. Co. Ltd. (KR) 2008-05-21 EP disclosed
US-20080096899-A1 N-Phenyl-2-Pyrimidine-Amine Derivatives and Process for the Preparation Thereof IL-YANG PHARM. CO., LTD. (KR) 2008-04-24 US disclosed
CN-101155786-A N-phenyl-2-pyrimidine-amine derivatives and process for the preparation thereof IL YANG PHARM CO LTD (KR) 2008-04-02 CN disclosed
US-20070213330-A1 Anticancer agents; antiproliferative agents METHYLGENE INC. (CA) 2007-09-13 US disclosed
US-20070213330-A1 Anticancer agents; antiproliferative agents METHYLGENE INC. (CA) 2007-09-13 US disclosed
US-7253204-B2 Antiproliferative agents METHYLGENE INC. (CA) 2007-08-07 US disclosed
WO-2007018325-A1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF IL-YANG PHARM. CO., LTD. (KR) 2007-02-15 WO disclosed
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed
EP-0233461-B1 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 1996-03-20 EP disclosed
US-4876252-A ADMINISTERING ANTIASTHMATIC OR ANTIALLERGEN AMERICAN CYANAMID COMPANY (US) 1989-10-24 US disclosed
US-4788195-A TREATING ASTHMA, ALLERGIC DISEASES, INFLAMMATION AND DIABETES IN MAMMALS AMERICAN CYANAMID COMPANY (US) 1988-11-29 US disclosed
EP-0233461-A2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID COMPANY (US) 1987-08-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213330-A1 Anticancer agents; antiproliferative agents HDAC1, HDAC11, HDAC5 ABL1 1137/4885BCR 2721/4885PRKCA 1179/4885
US-20080096899-A1 N-Phenyl-2-Pyrimidine-Amine Derivatives and Process for the Preparation Thereof ITPA, TYMP, THPO ABL1 451/4885BCR 990/4885PRKCA 3167/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.