SCHEMBL21032222

SCHEMBL21032222

O=S1(=O)C=C(I)c2cnccc21

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CDC25B P30305 1/20 0.33
IMPDH2 P12268 2/20 0.32
IMPDH1 P20839 2/20 0.32
EP300 Q09472 1/20 0.32
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21266565 0.77 CA1 (0.41) PTGDR2MAOAMAOBCDC25BIMPDH2
SCHEMBL21032218 0.71 GPR3 (0.46) MAOBIMPDH2IMPDH1EP300
SCHEMBL21157146 0.70 GPR3 (0.44) MAOAMAOBCDC25B
SCHEMBL21917575 0.67 EGFR (0.38) MAOAMAOBCDC25BIMPDH2IMPDH1
SCHEMBL8229992 0.66 PTGDR2 (0.33) PTGDR2
SCHEMBL18818680 0.65 CDC25B (0.32) CDC25B
SCHEMBL8285749 0.61 LMNA (0.39) MAOAMAOBCDC25B
SCHEMBL21032156 0.61 VEGFA (0.40) MAOAMAOBCDC25B
SCHEMBL21157145 0.61 GPR3 (0.44) MAOAMAOBCDC25B
SCHEMBL22827924 0.60 MAOA (0.37) MAOAMAOBCDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed