SCHEMBL21034056

SCHEMBL21034056

COC(=O)c1ccccc1OS(=O)(=O)F

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.67
SLC6A3 Q01959 3/20 0.54
SLC6A4 P31645 2/20 0.53
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA5A P35218 1/20 0.51
CA9 Q16790 1/20 0.51
TSHR P16473 2/20 0.50
LMNA P02545 1/20 0.50
HSD17B10 Q99714 2/20 0.49
ALDH1A1 P00352 2/20 0.49
ELANE P08246 1/20 0.49
CFTR P13569 1/20 0.49
KMT2A Q03164 3/20 0.48
HTT P42858 1/20 0.48
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
ATM Q13315 1/20 0.47
MAPT P10636 3/20 0.47
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27480641 0.84 L3MBTL1 (0.69) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL648371 0.84 L3MBTL1 (0.69) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL32665166 0.82 ELANE (0.52) L3MBTL1TSHRLMNAHSD17B10ALDH1A1
SCHEMBL4442981 0.82 L3MBTL1 (0.61) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL8606486 0.81 L3MBTL1 (0.65) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL7113435 0.81 L3MBTL1 (0.65) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL19122203 0.80 ELANE (0.53) TSHRLMNAHSD17B10ALDH1A1ELANE
SCHEMBL1665977 0.80 MAPT (0.70) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL3529817 0.80 L3MBTL1 (1.00) L3MBTL1SLC6A3SLC6A4CA1CA2
SCHEMBL28176283 0.80 SLC6A3 (0.62) L3MBTL1SLC6A3SLC6A4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3715342-B1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF ZHONGHONGXIN INVEST HOLDINGS SHENZHEN CO LTD (CN) 2024-08-07 EP disclosed
US-11091442-B2 Fluorosulfonyl-containing compound, intermediate thereof, preparation method therefor and use thereof SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2021-08-17 US disclosed
US-11091442-B2 Fluorosulfonyl-containing compound, intermediate thereof, preparation method therefor and use thereof SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2021-08-17 US disclosed
US-11046653-B2 2021-06-29 US disclosed
US-11046653-B2 2021-06-29 US disclosed
US-20200369619-A1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2020-11-26 US disclosed
US-20200369619-A1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2020-11-26 US disclosed
EP-3715342-A1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2020-09-30 EP disclosed
EP-3715342-A1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2020-09-30 EP disclosed
CN-110590609-A Fluorine-containing sulfonyl compound, intermediate, preparation method and application thereof 中国科学院上海有机化学研究所 2019-12-20 CN disclosed
WO-2019101132-A1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海有机化学研究所 2019-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11046653-B2 CYP4F11, NOTUM, CYP2F1 L3MBTL1 3471/4885SLC6A3 437/4885SLC6A4 182/4885
US-20200369619-A1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF WEE1, NOTUM, WEE2 L3MBTL1 1956/4885SLC6A3 966/4885SLC6A4 330/4885
US-11091442-B2 Fluorosulfonyl-containing compound, intermediate thereof, preparation method therefor and use thereof WEE1, NOTUM, WEE2 L3MBTL1 1956/4885SLC6A3 966/4885SLC6A4 330/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.