SCHEMBL21034935

SCHEMBL21034935

CC(C)(C)OC(=O)NC1CCN(C(=O)[C@@H]2CN(Cc3ccc(C(F)(F)F)cc3)CCN2S(=O)(=O)c2ccc3cc(OC4CCCC4)ccc3c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 4/20 0.42
DRD4 P21917 1/20 0.39
ADRB2 P07550 1/20 0.39
ROCK2 O75116 1/20 0.39
SCN9A Q15858 1/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
MCHR1 Q99705 2/20 0.38
KCNH2 Q12809 1/20 0.38
MLNR O43193 1/20 0.38
WNT3 P56703 3/20 0.37
SFRP1 Q8N474 3/20 0.37
PRKAA2 P54646 1/20 0.37
RORC P51449 2/20 0.37
TEAD1 P28347 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21035072 0.91 CCR4 (0.42) CCR4ROCK2MMP1MMP3MMP7
SCHEMBL21035343 0.91 CCR4 (0.42) CCR4ROCK2MMP1MMP3MMP7
SCHEMBL21035330 0.91 CCR4 (0.42) CCR4ROCK2MMP1MMP3MMP7
SCHEMBL21036254 0.91 CCR4 (0.40) CCR4ROCK2MMP1MMP3MMP7
SCHEMBL21035452 0.91 CCR4 (0.40) CCR4ROCK2MMP1MMP3MMP7
SCHEMBL21034971 0.88 ADRB2 (0.38) CCR4DRD4ADRB2ROCK2SCN9A
SCHEMBL21035477 0.87 ADRB2 (0.43) CCR4ADRB2SCN9AMMP1MMP3
SCHEMBL21034936 0.87 ADRB2 (0.43) CCR4ADRB2SCN9AMMP1MMP3
SCHEMBL21035481 0.87 ADRB2 (0.43) CCR4ADRB2SCN9AMMP1MMP3
SCHEMBL21035570 0.85 MMP1 (0.40) SCN9AMMP1MMP3MMP7MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed