SCHEMBL21035452

SCHEMBL21035452

CC(C)(C)OC(=O)NC1CCN(C(=O)[C@@H]2CN(Cc3ccc(C4(C(F)(F)F)CC4)cc3)CCN2S(=O)(=O)c2ccc3cc(OC4CCCC4)ccc3c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 4/20 0.40
ROCK2 O75116 2/20 0.38
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
MMP1 P03956 4/20 0.36
MMP13 P45452 4/20 0.36
MMP9 P14780 3/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
PRKAA2 P54646 4/20 0.35
WNT3 P56703 3/20 0.34
SFRP1 Q8N474 3/20 0.34
ADAM17 P78536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21036254 1.00 CCR4 (0.40) CCR4ROCK2PARP1PARP2MMP1
SCHEMBL21034935 0.91 CCR4 (0.42) CCR4ROCK2MMP1MMP13MMP9
SCHEMBL21035343 0.88 CCR4 (0.42) CCR4ROCK2PARP1PARP2MMP1
SCHEMBL21035330 0.88 CCR4 (0.42) CCR4ROCK2PARP1PARP2MMP1
SCHEMBL21035072 0.88 CCR4 (0.42) CCR4ROCK2PARP1PARP2MMP1
SCHEMBL21002090 0.88 MMP1 (0.37) CCR4ROCK2MMP1MMP13MMP9
SCHEMBL21002092 0.88 MMP1 (0.37) CCR4ROCK2MMP1MMP13MMP9
SCHEMBL21035486 0.87 MMP13 (0.39) CCR4MMP1MMP13MMP9MMP3
SCHEMBL21036241 0.87 MMP13 (0.39) CCR4MMP1MMP13MMP9MMP3
SCHEMBL21036224 0.86 GHSR (0.41) CCR4MMP1MMP13MMP9MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed