SCHEMBL21035508

SCHEMBL21035508

CC(C)(C)OC(=O)NC1CCN(C(=O)[C@@H]2CN(Cc3ccc(-c4ccc(C(F)(F)F)cc4)nc3)CCN2S(=O)(=O)c2ccc(OCC3CCCCC3)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.41
KCNQ1 P51787 1/20 0.39
GPR119 Q8TDV5 3/20 0.39
MMP1 P03956 6/20 0.37
MMP13 P45452 5/20 0.37
ADAM17 P78536 4/20 0.37
MMP9 P14780 3/20 0.37
SLC6A5 Q9Y345 2/20 0.37
HDAC1 Q13547 1/20 0.37
MMP3 P08254 1/20 0.35
MMP7 P09237 1/20 0.35
NAMPT P43490 1/20 0.35
STAT3 P40763 2/20 0.35
CHRNA7 P36544 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21035636 0.94 GPR119 (0.39) SCN9AGPR119MMP1MMP13ADAM17
SCHEMBL21035641 0.94 GPR119 (0.39) KCNQ1GPR119MMP1MMP13ADAM17
SCHEMBL21035604 0.94 SCN9A (0.39) SCN9AKCNQ1MMP1MMP13ADAM17
SCHEMBL21035570 0.93 MMP1 (0.40) SCN9AMMP1MMP13ADAM17MMP9
SCHEMBL21036229 0.93 GPR119 (0.39) KCNQ1GPR119MMP1MMP13ADAM17
SCHEMBL21034960 0.92 GPR119 (0.40) SCN9AGPR119MMP1MMP13ADAM17
SCHEMBL21034973 0.92 GPR119 (0.39) KCNQ1GPR119MMP1MMP13ADAM17
SCHEMBL21035090 0.91 GPR119 (0.40) KCNQ1GPR119MMP1MMP13ADAM17
SCHEMBL21035530 0.89 MMP1 (0.39) MMP1MMP13ADAM17MMP9MMP3
SCHEMBL21035509 0.88 KCNQ1 (0.40) KCNQ1MMP1MMP13ADAM17MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed